Epigenetics probes


Target Probe Control Targeted domain Mode of action Recommended concentration Target origin
EP300, CREBBP A-485 A-486 HAT domain Inhibitor 0.8 µM human
BRD7, BRD9 VZ185 cisVZ185 PROTAC degrader 300 nM human
SMARCA2, SMARCA4 FHT-2344 FHT-5908 Inhibitor ≤ 1 µM human
BRD2, BRD3, BRD4, BRDT GSK046 no record.controls BD2 Inhibitor ≤ 10 µM human
BRD2, BRD3, BRD4, BRDT GSK620 no record.controls BD2 Inhibitor ≤ 10 µM human
BRD2, BRD3, BRD4, BRDT GSK778 no record.controls BD1 Inhibitor ≤ 1 µM human
BRD2, BRD3, BRD4, BRDT GSK789 GSK791 BD1 Inhibitor ≤ 10 µM human
BRD2, BRD3, BRD4, BRDT GSK973 GSK943 BD2 Inhibitor ≤ 10 µM human
KAT6A, KAT6B WM-1119 WM-2474 AcCoA binding site Inhibitor 1 µM (≤ 10 µM) human