| Target | Probe | Control | Targeted domain | Mode of action | Recommended concentration | Target origin |
|---|---|---|---|---|---|---|
| EP300, CREBBP | A-485 | A-486 | HAT domain | Inhibitor | 0.8 µM | human |
| BRD7, BRD9 | VZ185 | cisVZ185 | — | PROTAC degrader | 300 nM | human |
| SMARCA2, SMARCA4 | FHT-2344 | FHT-5908 | — | Inhibitor | ≤ 1 µM | human |
| BRD2, BRD3, BRD4, BRDT | GSK046 | no record.controls | BD2 | Inhibitor | ≤ 10 µM | human |
| BRD2, BRD3, BRD4, BRDT | GSK620 | no record.controls | BD2 | Inhibitor | ≤ 10 µM | human |
| BRD2, BRD3, BRD4, BRDT | GSK778 | no record.controls | BD1 | Inhibitor | ≤ 1 µM | human |
| BRD2, BRD3, BRD4, BRDT | GSK789 | GSK791 | BD1 | Inhibitor | ≤ 10 µM | human |
| BRD2, BRD3, BRD4, BRDT | GSK973 | GSK943 | BD2 | Inhibitor | ≤ 10 µM | human |
| KAT6A, KAT6B | WM-1119 | WM-2474 | AcCoA binding site | Inhibitor | 1 µM (≤ 10 µM) | human |