Other targets probes


Target Probe Control Targeted domain Mode of action Recommended concentration Target origin
BCL2L1 A-1155463 A-1107969 BCL domain Inhibitor ≤ 5 µM human
BCL2 A-1211212 A-1210227 Inhibitor ≤ 5 µM human
NR3C1 BI 653048 BI-3047 Ligand binding domain Agonist 1 µM human
ITGAL BI-1950 BI-9446 I-domain Inhibitor 100 nM human
BCL6 BI-3802 BI-5273 BTB/POZ, binds at interface of 2 monomers Degrader ≤ 1 µM human
BCL6 BI-3812 BI-5273 BTB/POZ, binds at interface of 2 monomers Inhibitor ≤ 1 µM human
BCL6 CCT369260 CCT393732 BTB domain Degrader ≤ 1 µM human
MCL1 JNJ-4355 JNJ-78732576 BCL domain Inhibitor ≤ 10 µM human
NRLP3 JNJ-79883960 JNJ-78832000 NACHT domain Inhibitor ≤ 10 µM human
RORC JNJ-54119936 JNJ-53721590 Orthosteric site of binding domain Inverse agonist ≤ 1 µM human
RXRA, RXRB, RXRG JP3000 JP3001 Ligand binding domain Agonist 0.1 - 1 µM human
SLC16A3 MSC-4381 MSC-0516 Inhibitor ≤ 10 µM human
BCL6 TP-021 TP-021n Bric-a-brac (BTB) domain Inhibitor 1 -10 µM human