| BCL2L1 |
A-1155463 |
A-1107969 |
BCL domain |
Inhibitor |
≤ 5 µM |
human |
| BCL2 |
A-1211212 |
A-1210227 |
— |
Inhibitor |
≤ 5 µM |
human |
| NR3C1 |
BI 653048 |
BI-3047 |
Ligand binding domain |
Agonist |
1 µM |
human |
| ITGAL |
BI-1950 |
BI-9446 |
I-domain |
Inhibitor |
100 nM |
human |
| BCL6 |
BI-3802 |
BI-5273 |
BTB/POZ, binds at interface of 2 monomers |
Degrader |
≤ 1 µM |
human |
| BCL6 |
BI-3812 |
BI-5273 |
BTB/POZ, binds at interface of 2 monomers |
Inhibitor |
≤ 1 µM |
human |
| BCL6 |
CCT369260 |
CCT393732 |
BTB domain |
Degrader |
≤ 1 µM |
human |
| MCL1 |
JNJ-4355 |
JNJ-78732576 |
BCL domain |
Inhibitor |
≤ 10 µM |
human |
| NRLP3 |
JNJ-79883960 |
JNJ-78832000 |
NACHT domain |
Inhibitor |
≤ 10 µM |
human |
| RORC |
JNJ-54119936 |
JNJ-53721590 |
Orthosteric site of binding domain |
Inverse agonist |
≤ 1 µM |
human |
| RXRA, RXRB, RXRG |
JP3000 |
JP3001 |
Ligand binding domain |
Agonist |
0.1 - 1 µM |
human |
| SLC16A3 |
MSC-4381 |
MSC-0516 |
— |
Inhibitor |
≤ 10 µM |
human |
| BCL6 |
TP-021 |
TP-021n |
Bric-a-brac (BTB) domain |
Inhibitor |
1 -10 µM |
human |