| Target | Probe | Control | Targeted domain | Mode of action | Recommended concentration | Target origin |
|---|---|---|---|---|---|---|
| BCL2L1 | A-1155463 | A-1107969 | BCL domain | Inhibitor | ≤ 5 µM | human |
| BCL2 | A-1211212 | A-1210227 | — | Inhibitor | ≤ 5 µM | human |
| NR3C1 | BI 653048 | BI-3047 | Ligand binding domain | Agonist | 1 µM | human |
| ITGAL | BI-1950 | BI-9446 | I-domain | Inhibitor | 100 nM | human |
| BCL6 | BI-3802 | BI-5273 | BTB/POZ, binds at interface of 2 monomers | Degrader | ≤ 1 µM | human |
| BCL6 | BI-3812 | BI-5273 | BTB/POZ, binds at interface of 2 monomers | Inhibitor | ≤ 1 µM | human |
| BCL6 | CCT369260 | CCT393732 | BTB domain | Degrader | ≤ 1 µM | human |
| MCL1 | JNJ-4355 | JNJ-78732576 | BCL domain | Inhibitor | ≤ 10 µM | human |
| NRLP3 | JNJ-79883960 | JNJ-78832000 | NACHT domain | Inhibitor | ≤ 10 µM | human |
| RORC | JNJ-54119936 | JNJ-53721590 | Orthosteric site of binding domain | Inverse agonist | ≤ 1 µM | human |
| RXRA, RXRB, RXRG | JP3000 | JP3001 | Ligand binding domain | Agonist | 0.1 - 1 µM | human |
| SLC16A3 | MSC-4381 | MSC-0516 | — | Inhibitor | ≤ 10 µM | human |
| BCL6 | TP-021 | TP-021n | Bric-a-brac (BTB) domain | Inhibitor | 1 -10 µM | human |