Target	Probe	Control	Targeted domain	Mode of action	Recommended concentration	Target origin
CFTR	A-1596586	A-1596584	—	Corrector	≤ 1 µM	human
TRPA1	A-079	A-226	—	Antagonist	1 µM	human
P2RX4	BAY-1797	BAY-207	—	Inhibitor	0.1 - 1 µM	human
TRPA1	BAY-390	BAY-9897	—	Inhibitor	100 nM	human
Epithelial sodium channel	BI-8668	BI-0337	—	Inhibitor	1 µM	human
SLC9A1	BI-9627	BI-0054	—	Antagonist	≤ 5 µM	human
GRIN2A	JNJ-78911118	JNJ-77914993	GRIN1/GRIN2A interface	Negative Allosteric Modulator	≤ 10 µM	human
TRPM8	PF-05105679	PF-05257137	—	Antagonist	1 µM	human
GABRA5	RO4938581	RO4991571	—	Negative allosteric modulator	≤ 1 µM	human
HCN1	RO-275	RO7239047	—	Suppressor	1 µM	human
GRIN2A	TP-050	TP-050n	GRIN1/GRIN2A ligand binding domain (Tyr 144)	Positive allosteric modulator	≤ 30 µM	human