Potency data for probe BAY-899 and control BAY-897
No in vitro potency data available.
In cell potency
| Target name | Target information | Species | Assay description | BAY-899 | BAY-897 | Publication of assay conditions |
|---|---|---|---|---|---|---|
| LHCGR | Homo sapiens | Cell-based assay (LH Antagonism) | IC50 = 185 nM | PMID: 31670515 | ||
| FSHR | Homo sapiens | Cell-based assay (FSH Antagonism) | IC50 > 16 µM | PMID: 31670515 | ||
| TSHR | Homo sapiens | Cell-based assay (TSH Antagonism) | IC50 = 24 µM | PMID: 31670515 | ||
| LHCGR | Homo sapiens | Cell-based assay (LH Antagonism) | IC50 > 16 µM | |||
| FSHR | Homo sapiens | Cell-based assay (FSH Antagonism) | IC50 > 16 µM |