Potency data for probe (R)-ZINC-3573 and control (S)-ZINC-3573
No in vitro potency data available.
In cell potency
| Target name | Target information | Species | Assay description | (R)-ZINC-3573 | (S)-ZINC-3573 | Publication of assay conditions |
|---|---|---|---|---|---|---|
| MRGPRX2 | Homo sapiens | PRESTO-Tango concentration response assay | EC50 = 740 nM (n=4) | EC50 > 100 µM (n=4) | PMID: 28288109 | |
| MRGPRX2 | Homo sapiens | FLIPR assay | EC50 = 1 µM (n=5) | EC50 > 100 µM (n=5) | PMID: 28288109 |