Potency data for probe BAY-7598 and control BAY-694
In vitro potency
| Target name | Target information | Species | Assay description | BAY-7598 | BAY-694 | Publication of assay conditions |
|---|---|---|---|---|---|---|
| MMP12 | Homo sapiens | Biochemical assay (MMP12) | IC50 = 0.085 nM | IC50 = 80 nM | ||
| MMP12 | Homo sapiens | Biophysical assay (SPR biosensor-based assay) | Kd = 0.004 nM |
No in cell potency data available.