Potency data for probe BI-1935 and control BI-2049
In vitro potency
| Target name | Target information | Species | Assay description | BI-1935 | BI-2049 | Publication of assay conditions |
|---|---|---|---|---|---|---|
| EPHX2 | Homo sapiens | Human soluble epoxide hydrolase inhibition | IC50 = 7 nM | IC50 > 3 µM |
In cell potency
| Target name | Target information | Species | Assay description | BI-1935 | BI-2049 | Publication of assay conditions |
|---|---|---|---|---|---|---|
| EPHX2 | Homo sapiens | Cellular assay: Human Hep G2 Cells, ELISA readout | IC50 < 1 nM |