Potency data for probe MSD-CYP11B2 and control MSD-CYP11B2 Negative control
In vitro potency
| Target name | Target information | Species | Assay description | Compound conc. | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|---|
| ADRA2B | Homo sapiens | Panlabs assay (ADRA2B) | 10 µM | IC50 = 4.700 µM | |||
| HTR2B | Homo sapiens | Panlabs assay (HTR2B) | 10 µM | IC50 = 5.330 µM | |||
| ADRB1 | Homo sapiens | Panlabs assay (ADRB1) | 10 µM | IC50 = 9.620 µM |
In cell potency
| Target name | Target information | Species | Assay description | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|
| CYP11B2 | V79 cell lines stably expressing human CYP11B2 enzyme | Homo sapiens | Assay using V79 cell lines (CYP11B2) | IC50 = 2.300 nM | IC50 > 10 µM | PMID: 26005536 |
| CYP11B1 | V79 cell lines stably expressing human CYP11B1 enzyme | Homo sapiens | Assay using V79 cell lines (CYP11B1) | IC50 = 142 nM | IC50 > 10 µM | PMID: 26005536 |