Potency data for probe TP-051 and control TP-051n
In vitro potency
| Target name | Target information | Species | Assay description | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|
| FFAR1 | Membrane fraction prepared from CHO cells expressing human FFAR1 | Homo sapiens | FFAR1 binding assay | Ki = 16 nM | Ki > 10 µM | PMID: 22428944 |
In cell potency
| Target name | Target information | Species | Assay description | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|
| FFAR1 | CHO cells expressing human FFAR1 | Homo sapiens | FLIPR functional assay (Ca influx activity of CHO cells) | EC50 = 25 nM | EC50 > 10 µM | PMID: 22428944 |