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Selectivity data for probe C3TD879 and control C3TD879-N


Coming soon

C3TD879

The panel was screened at an ATP conc. of 1 µM.

Conclusion: C3TD879 shows > 75-fold selectivity over every human kinase except for AAK1 (17-fold) .

Target protein HGNC name Species % activity at 1 µM
AAK1(h) AAK1 Homo sapiens 13.0
Abl(h) ABL1 Homo sapiens 99.0
ACK1(h) TNK2 Homo sapiens 39.0
ACTR2(h) ACTR2 Homo sapiens 96.0
ALK(h) ALK Homo sapiens 77.0
ALK1(h) ACVRL1 Homo sapiens 94.0
ALK2(h) ACVR1 Homo sapiens 122.0
ALK4(h) ACVR1B Homo sapiens 94.0
ALK6(h) BMPR1B Homo sapiens 74.0
AMPKalpha1(h) PRKAA1 Homo sapiens 120.0
AMPKalpha2(h) PRKAA2 Homo sapiens 117.0
A-Raf(h) ARAF Homo sapiens 97.0
Arg(h) ABL2 Homo sapiens 72.0
ARK5(h) NUAK1 Homo sapiens 85.0
ASK1(h) MAP3K5 Homo sapiens 100.0
ATM(h) ATM Homo sapiens 103.0
ATR/ATRIP(h) ATR
ATRIP
Homo sapiens 110.0
Aurora-A(h) AURKA Homo sapiens 97.0
Aurora-B(h) AURKB Homo sapiens 109.0
Aurora-C(h) AURKC Homo sapiens 94.0
Axl(h) AXL Homo sapiens 91.0
BIKE(h) BMP2K Homo sapiens 50.0
Blk(h) BLK Homo sapiens 88.0
BMPR2(h) BMPR2 Homo sapiens 85.0
Bmx(h) BMX Homo sapiens 97.0
B-Raf(h) BRAF Homo sapiens 110.0
BRK(h) PTK6 Homo sapiens 83.0
BrSK1(h) BRSK1 Homo sapiens 96.0
BrSK2(h) BRSK2 Homo sapiens 83.0
BTK(h) BTK Homo sapiens 122.0
CaMKI(h) CAMK1 Homo sapiens 104.0
CaMKIIalpha(h) CAMK2A Homo sapiens 88.0
CaMKIIbeta(h) CAMK2B Homo sapiens 93.0
CaMKIIgamma(h) CAMK2G Homo sapiens 106.0
CaMKIIdelta(h) CAMK2D Homo sapiens 96.0
CaMKIbeta(h) PNCK Homo sapiens 85.0
CaMKIV(h) CAMK4 Homo sapiens 99.0
CaMKIgamma(h) CAMK1G Homo sapiens 110.0
CaMKIdelta(h) CAMK1D Homo sapiens 89.0
CaMKK1(h) CAMKK1 Homo sapiens 89.0
CaMKK2(h) CAMKK2 Homo sapiens 96.0
Cdc7/cyclinB1(h) CDC7
CCNB1
Homo sapiens 75.0
CDK1/cyclinB(h) CDK1
CCNB1
Homo sapiens 94.0
CDK12/cyclinK(h) CDK12
CCNK
Homo sapiens 89.0
CDK13/cyclinK(h) CDK13
CCNK
Homo sapiens 99.0
CDK14/cyclinY(h) CDK14
CCNY
Homo sapiens 91.0
CDK16/cyclinY(h) CDK16
CCNY
Homo sapiens 98.0
CDK17/cyclinY(h) CDK17
CCNY
Homo sapiens 108.0
CDK18/cyclinY(h) CDK18
CCNY
Homo sapiens 94.0
CDK2/cyclinA(h) CDK2
CCNA2
Homo sapiens 87.0
CDK2/cyclinE(h) CDK2
CCNE1
Homo sapiens 92.0
CDK3/cyclinE(h) CDK3
CCNE1
Homo sapiens 102.0
CDK4/cyclinD3(h) CDK4
CCND3
Homo sapiens 74.0
CDK5/p25(h) CDK5
CDK5R1
Homo sapiens 72.0
CDK5/p35(h) CDK5
CDK5R1
Homo sapiens 79.0
CDK6/cyclinD3(h) CDK6
CCND3
Homo sapiens 90.0
CDK7/cyclinH/MAT1(h) CDK7
CCNH
MNAT1
Homo sapiens 95.0
CDK9/cyclin T1(h) CDK9
CCNT1
Homo sapiens 81.0
CDKL1(h) CDKL1 Homo sapiens 99.0
CDKL2(h) CDKL2 Homo sapiens 80.0
CDKL3(h) CDKL3 Homo sapiens 79.0
CDKL4(h) CDKL4 Homo sapiens 104.0
ChaK1(h) TRPM7 Homo sapiens 106.0
CHK1(h) CHEK1 Homo sapiens 108.0
CHK2(h) CHEK2 Homo sapiens 95.0
CK1alpha(h) CSNK1A1 Homo sapiens 97.0
CK1gamma1(h) CSNK1G1 Homo sapiens 101.0
CK1gamma2(h) CSNK1G2 Homo sapiens 97.0
CK1gamma3(h) CSNK1G3 Homo sapiens 84.0
CK1delta(h) CSNK1D Homo sapiens 96.0
CK1epsilon(h) CSNK1E Homo sapiens 96.0
CK2(h) Homo sapiens 112.0
CK2alpha1(h) CSNK2A1 Homo sapiens 112.0
CK2alpha2(h) CSNK2A2 Homo sapiens 115.0
cKit(h) KIT Homo sapiens 85.0
CLIK1(h) STK35 Homo sapiens 97.0
CLK1(h) CLK1 Homo sapiens 88.0
CLK2(h) CLK2 Homo sapiens 106.0
CLK3(h) CLK3 Homo sapiens 107.0
CLK4(h) CLK4 Homo sapiens 85.0
c-RAF(h) RAF1 Homo sapiens 106.0
CRIK(h) aka CITK CIT Homo sapiens 0.0
CSK(h) CSK Homo sapiens 92.0
cSRC(h) SRC Homo sapiens 93.0
DAPK1(h) DAPK1 Homo sapiens 82.0
DAPK2(h) DAPK2 Homo sapiens 109.0
DCAMKL1(h) DCLK1 Homo sapiens 95.0
DCAMKL2(h) DCLK2 Homo sapiens 104.0
DCAMKL3(h) DCLK3 Homo sapiens 86.0
DDR1(h) DDR1 Homo sapiens 98.0
DDR2(h) DDR2 Homo sapiens 85.0
DMPK(h) DMPK Homo sapiens 93.0
DNA-PK(h) PRKDC Homo sapiens 107.0
DRAK1(h) STK17A Homo sapiens 80.0
DRAK2(h) STK17B Homo sapiens 50.0
DYRK1A(h) DYRK1A Homo sapiens 112.0
DYRK1B(h) DYRK1B Homo sapiens 108.0
DYRK2(h) DYRK2 Homo sapiens 101.0
DYRK3(h) DYRK3 Homo sapiens 99.0
eEF-2K(h) EEF2K Homo sapiens 92.0
EGFR(h) EGFR Homo sapiens 107.0
EphA1(h) EPHA1 Homo sapiens 92.0
EphA2(h) EPHA2 Homo sapiens 95.0
EphA3(h) EPHA3 Homo sapiens 79.0
EphA4(h) EPHA4 Homo sapiens 92.0
EphA5(h) EPHA5 Homo sapiens 89.0
EphA7(h) EPHA7 Homo sapiens 114.0
EphA8(h) EPHA8 Homo sapiens 115.0
EphB1(h) EPHB1 Homo sapiens 83.0
EphB2(h) EPHB2 Homo sapiens 96.0
EphB3(h) EPHB3 Homo sapiens 79.0
EphB4(h) EPHB4 Homo sapiens 107.0
ErbB2(h) ERBB2 Homo sapiens 97.0
ErbB4(h) ERBB4 Homo sapiens 94.0
FAK(h) PTK2 Homo sapiens 96.0
Fer(h) FER Homo sapiens 103.0
Fes(h) FES Homo sapiens 111.0
FGFR1(h) FGFR1 Homo sapiens 100.0
FGFR2(h) FGFR2 Homo sapiens 89.0
FGFR3(h) FGFR3 Homo sapiens 86.0
FGFR4(h) FGFR4 Homo sapiens 114.0
Fgr(h) FGR Homo sapiens 97.0
Flt1(h) FLT1 Homo sapiens 125.0
Flt3(h) FLT3 Homo sapiens 84.0
Flt4(h) FLT4 Homo sapiens 96.0
Fms(h) CSF1R Homo sapiens 115.0
Fyn(h) FYN Homo sapiens 100.0
GCK(h) GCK Homo sapiens 118.0
GCN2(h) EIF2AK4 Homo sapiens 101.0
GRK1(h) GRK1 Homo sapiens 86.0
GRK2(h) GRK2 Homo sapiens 95.0
GRK3(h) GRK3 Homo sapiens 81.0
GRK5(h) GRK5 Homo sapiens 97.0
GRK6(h) GRK6 Homo sapiens 95.0
GRK7(h) GRK7 Homo sapiens 98.0
GSK3alpha(h) GSK3A Homo sapiens 87.0
GSK3beta(h) GSK3B Homo sapiens 93.0
Haspin(h) HASPIN Homo sapiens 140.0
Hck(h) HCK Homo sapiens 99.0
Hck(h) activated HCK Homo sapiens 111.0
HIPK1(h) HIPK1 Homo sapiens 100.0
HIPK2(h) HIPK2 Homo sapiens 105.0
HIPK3(h) HIPK3 Homo sapiens 85.0
HIPK4(h) HIPK4 Homo sapiens 52.0
HPK1(h) MAP4K1 Homo sapiens 73.0
HRI(h) EIF2AK1 Homo sapiens 80.0
ICK(h) CILK1 Homo sapiens 99.0
IGF-1R(h) IGF1R Homo sapiens 98.0
IGF-1R(h), activated IGF1R Homo sapiens 93.0
IKKalpha(h) CHUK Homo sapiens 98.0
IKKbeta(h) IKBKB Homo sapiens 99.0
IKKepsilon(h) IKBKE Homo sapiens 87.0
IR(h) INSR Homo sapiens 94.0
IR(h), activated INSR Homo sapiens 92.0
IRAK1(h) IRAK1 Homo sapiens 95.0
IRAK4(h) IRAK4 Homo sapiens 90.0
IRE1(h) ERN1 Homo sapiens 99.0
IRR(h) INSRR Homo sapiens 110.0
Itk(h) ITK Homo sapiens 86.0
JAK1(h) JAK1 Homo sapiens 85.0
JAK2(h) JAK2 Homo sapiens 104.0
JAK3(h) JAK3 Homo sapiens 106.0
JNK1alpha1(h) MAPK8 Homo sapiens 110.0
JNK2alpha2(h) MAPK9 Homo sapiens 99.0
JNK3(h) MAPK10 Homo sapiens 88.0
KDR(h) KDR Homo sapiens 78.0
LATS1(h) LATS1 Homo sapiens 90.0
LATS2(h) LATS2 Homo sapiens 102.0
Lck(h) LCK Homo sapiens 86.0
Lck(h) activated LCK Homo sapiens 119.0
LIMK1(h) LIMK1 Homo sapiens 70.0
LIMK2(h) LIMK2 Homo sapiens 72.0
LKB1(h) STK11 Homo sapiens 99.0
LOK(h) STK10 Homo sapiens 96.0
LRRK2(h) LRRK2 Homo sapiens 100.0
LTK(h) LTK Homo sapiens 97.0
Lyn(h) LYN Homo sapiens 80.0
MAK(h) MAK Homo sapiens 120.0
MAP4K3(h) MAP4K3 Homo sapiens 109.0
MAP4K4(h) MAP4K4 Homo sapiens 101.0
MAP4K5(h) MAP4K5 Homo sapiens 92.0
MAPK1(h) MAPK1 Homo sapiens 95.0
MAPKAP-K2(h) MAPKAPK2 Homo sapiens 72.0
MAPKAP-K3(h) MAPKAPK3 Homo sapiens 125.0
MARK1(h) MARK1 Homo sapiens 106.0
MARK3(h) MARK3 Homo sapiens 90.0
MARK4(h) MARK4 Homo sapiens 92.0
MEK1(h) MAP2K1 Homo sapiens 101.0
MEK2(h) MAP2K2 Homo sapiens 92.0
MEKK2(h) MAP3K2 Homo sapiens 122.0
MEKK3(h) MAP3K3 Homo sapiens 107.0
MELK(h) MELK Homo sapiens 82.0
Mer(h) MERTK Homo sapiens 105.0
Met(h) MET Homo sapiens 90.0
MINK(h) MINK1 Homo sapiens 89.0
MKK3(h) MAP2K3 Homo sapiens 97.0
MKK6(h) MAP2K6 Homo sapiens 101.0
MLCK(h) MYLK3 Homo sapiens 98.0
MLK1(h) MAP3K9 Homo sapiens 103.0
MLK2(h) MAP3K10 Homo sapiens 77.0
MLK3(h) MAP3K11 Homo sapiens 91.0
MLK4(h) MAP3K21 Homo sapiens 112.0
Mnk2(h) MKNK2 Homo sapiens 35.0
MOK(h) MOK Homo sapiens 90.0
MRCKalpha(h) CDC42BPA Homo sapiens 94.0
MRCKbeta(h) CDC42BPB Homo sapiens 100.0
MRCKgamma(h) CDC42BPG Homo sapiens 98.0
MSK1(h) RPS6KA5 Homo sapiens 111.0
MSK2(h) RPS6KA4 Homo sapiens 88.0
MSSK1(h) SRPK3 Homo sapiens 134.0
MST1(h) STK4 Homo sapiens 76.0
MST2(h) STK3 Homo sapiens 106.0
MST3(h) STK24 Homo sapiens 85.0
MST4(h) STK26 Homo sapiens 106.0
mTOR(h) MTOR Homo sapiens 95.0
mTOR/FKBP12(h) MTOR
FKBP1A
Homo sapiens 120.0
MuSK(h) MUSK Homo sapiens 96.0
MYLK2(h) MYLK2 Homo sapiens 76.0
MYO3B(h) MYO3B Homo sapiens 79.0
NDR1(h) STK38 Homo sapiens 100.0
NDR2(h) STK38L Homo sapiens 107.0
NEK1(h) NEK1 Homo sapiens 94.0
NEK11(h) NEK11 Homo sapiens 97.0
NEK2(h) NEK2 Homo sapiens 118.0
NEK3(h) NEK3 Homo sapiens 110.0
NEK4(h) NEK4 Homo sapiens 90.0
NEK6(h) NEK6 Homo sapiens 86.0
NEK7(h) NEK7 Homo sapiens 88.0
NEK9(h) NEK9 Homo sapiens 79.0
NIM1(h) NIM1K Homo sapiens 112.0
NLK(h) NLK Homo sapiens 98.0
NUAK2(h) NUAK2 Homo sapiens 72.0
OSR1(h) OXSR1 Homo sapiens 80.0
p70S6K(h) Homo sapiens 93.0
PAK1(h) PAK1 Homo sapiens 95.0
PAK2(h) PAK2 Homo sapiens 95.0
PAK3(h) PAK3 Homo sapiens 89.0
PAK4(h) PAK4 Homo sapiens 83.0
PAK5(h) PAK5 Homo sapiens 87.0
PAK6(h) PAK6 Homo sapiens 101.0
PAR-1Balpha(h) MARK2 Homo sapiens 88.0
PASK(h) PASK Homo sapiens 72.0
PDGFRalpha(h) PDGFRA Homo sapiens 116.0
PDGFRbeta(h) PDGFRB Homo sapiens 105.0
PDHK2(h) PDK2 Homo sapiens 87.0
PDHK4(h) PDK4 Homo sapiens 101.0
PDK1(h) PDK1 Homo sapiens 105.0
PEK(h) EIF2AK3 Homo sapiens 91.0
PhKgamma1(h) PHKG1 Homo sapiens 101.0
PhKgamma2(h) PHKG2 Homo sapiens 98.0
PI3 Kinase (p110alpha/p85alpha)(h) PIK3CA
PIK3R1
Homo sapiens 96.0
PI3 Kinase (p110beta/p85alpha)(h) PIK3CB
PIK3R1
Homo sapiens 102.0
PI3 Kinase (p110delta/p85alpha)(h) PIK3CD
PIK3R1
Homo sapiens 110.0
PI3 Kinase (p120gamma)(h) PIK3CG Homo sapiens 105.0
PI3KC2alpha(h) PIK3C2A Homo sapiens 102.0
PI3KC2gamma(h) PIK3C2G Homo sapiens 103.0
Pim-1(h) PIM1 Homo sapiens 95.0
Pim-2(h) PIM2 Homo sapiens 117.0
Pim-3(h) PIM3 Homo sapiens 103.0
PIP4K2alpha(h) PIP4K2A Homo sapiens 100.0
PIP5K1alpha(h) PIP5K1A Homo sapiens 103.0
PIP5K1gamma(h) PIP5K1C Homo sapiens 102.0
PKA(h) Homo sapiens 109.0
PKACbeta(h) PRKACB Homo sapiens 121.0
PKBalpha(h) AKT1 Homo sapiens 87.0
PKBbeta(h) AKT2 Homo sapiens 109.0
PKBgamma(h) AKT3 Homo sapiens 101.0
PKCalpha(h) PRKCA Homo sapiens 92.0
PKCbetaI(h) PRKCB Homo sapiens 90.0
PKCbetaII(h) PRKCB Homo sapiens 87.0
PKCgamma(h) PRKCG Homo sapiens 97.0
PKCdelta(h) PRKCD Homo sapiens 93.0
PKCepsilon(h) PRKCE Homo sapiens 97.0
PKCzeta(h) PRKCZ Homo sapiens 88.0
PKCeta(h) PRKCH Homo sapiens 118.0
PKCtheta(h) PRKCQ Homo sapiens 103.0
PKCiota(h) PRKCI Homo sapiens 110.0
PKCmu(h) PRKD1 Homo sapiens 109.0
PKD2(h) PRKD2 Homo sapiens 95.0
PKD3(h) PRKD3 Homo sapiens 97.0
PKG1beta(h) PRKG1 Homo sapiens 92.0
PKR(h) EIF2AK2 Homo sapiens 85.0
Plk1(h) PLK1 Homo sapiens 111.0
Plk3(h) PLK3 Homo sapiens 100.0
Plk4(h) PLK4 Homo sapiens 92.0
PRAK(h) MAPKAPK5 Homo sapiens 107.0
PRK1(h) PKN1 Homo sapiens 91.0
PRK2(h) PKN2 Homo sapiens 92.0
PRKG2(h) PRKG2 Homo sapiens 110.0
PrKX(h) PRKX Homo sapiens 101.0
PRP4(h) PRPF4B Homo sapiens 100.0
PTK5(h) FRK Homo sapiens 90.0
Pyk2(h) PTK2B Homo sapiens 76.0
Ret(h) RET Homo sapiens 97.0
RIPK1(h) RIPK1 Homo sapiens 84.0
RIPK2(h) RIPK2 Homo sapiens 97.0
ROCK-I(h) ROCK1 Homo sapiens 96.0
ROCK-II(h) ROCK2 Homo sapiens 96.0
Ron(h) MST1R Homo sapiens 111.0
Ros(h) ROS1 Homo sapiens 97.0
Rse(h) TYRO3 Homo sapiens 129.0
Rsk1(h) RPS6KA1 Homo sapiens 99.0
Rsk2(h) RPS6KA3 Homo sapiens 88.0
Rsk3(h) RPS6KA2 Homo sapiens 112.0
Rsk4(h) RPS6KA6 Homo sapiens 101.0
SAPK2a(h) MAPK14 Homo sapiens 94.0
SAPK2b(h) MAPK11 Homo sapiens 90.0
SAPK3(h) MAPK12 Homo sapiens 113.0
SAPK4(h) MAPK13 Homo sapiens 94.0
SBK1(h) SBK1 Homo sapiens 97.0
SGK(h) SGK1 Homo sapiens 113.0
SGK2(h) SGK2 Homo sapiens 82.0
SGK3(h) SGK3 Homo sapiens 102.0
SIK(h) SIK1 Homo sapiens 105.0
SIK2(h) SIK2 Homo sapiens 109.0
SIK3(h) SIK3 Homo sapiens 105.0
SLK(h) SLK Homo sapiens 109.0
Snk(h) PLK2 Homo sapiens 94.0
SNRK(h) SNRK Homo sapiens 111.0
SRMS(h) SRMS Homo sapiens 86.0
SRPK1(h) SRPK1 Homo sapiens 95.0
SRPK2(h) SRPK2 Homo sapiens 93.0
STK16(h) STK16 Homo sapiens 94.0
STK25(h) STK25 Homo sapiens 92.0
STK32A(h) STK32A Homo sapiens 90.0
STK32B(h) STK32B Homo sapiens 115.0
STK32C(h) STK32C Homo sapiens 85.0
STK33(h) STK33 Homo sapiens 98.0
STK39(h) STK39 Homo sapiens 102.0
Syk(h) SYK Homo sapiens 66.0
TAF1L(h) TAF1L Homo sapiens 101.0
TAK1(h) MAP3K7 Homo sapiens 91.0
TAO1(h) TAOK1 Homo sapiens 83.0
TAO2(h) TAOK2 Homo sapiens 90.0
TAO3(h) TAOK3 Homo sapiens 100.0
TBK1(h) TBK1 Homo sapiens 100.0
Tec(h) activated TEC Homo sapiens 126.0
TGFBR1(h) TGFBR1 Homo sapiens 103.0
TGFBR2(h) TGFBR2 Homo sapiens 96.0
Tie2(h) TEK Homo sapiens 99.0
TLK1(h) TLK1 Homo sapiens 82.0
TLK2(h) TLK2 Homo sapiens 92.0
TNIK(h) TNIK Homo sapiens 93.0
TRB2(h) TRIB2 Homo sapiens 104.0
TrkA(h) NTRK1 Homo sapiens 105.0
TrkB(h) NTRK2 Homo sapiens 84.0
TrkC(h) NTRK3 Homo sapiens 86.0
TSSK1(h) TSSK1B Homo sapiens 116.0
TSSK2(h) TSSK2 Homo sapiens 113.0
TSSK3(h) TSSK3 Homo sapiens 96.0
TSSK4(h) TSSK4 Homo sapiens 117.0
TTBK1(h) TTBK1 Homo sapiens 96.0
TTBK2(h) TTBK2 Homo sapiens 94.0
TTK(h) TTK Homo sapiens 102.0
Txk(h) TXK Homo sapiens 110.0
TYK2(h) TYK2 Homo sapiens 103.0
ULK1(h) ULK1 Homo sapiens 95.0
ULK2(h) ULK2 Homo sapiens 98.0
ULK3(h) ULK3 Homo sapiens 95.0
VRK1(h) VRK1 Homo sapiens 99.0
VRK2(h) VRK2 Homo sapiens 100.0
Wee1(h) WEE1 Homo sapiens 94.0
Wee1B(h) WEE2 Homo sapiens 88.0
WNK1(h) WNK1 Homo sapiens 109.0
WNK2(h) WNK2 Homo sapiens 94.0
WNK3(h) WNK3 Homo sapiens 85.0
WNK4(h) WNK4 Homo sapiens 97.0
Yes(h) YES1 Homo sapiens 87.0
ZAK(h) MAP3K20 Homo sapiens 83.0
ZAP-70(h) ZAP70 Homo sapiens 71.0
ZIPK(h) DAPK3 Homo sapiens 94.0