Selectivity data for probe T-10430 and control T-10404
Coming soon
T-10430
For the Ca2+ aequorin assay the GPCR plasmids from the PrestoTango panel were utilized and 1 µM compound was used. The assay was performed from Mohamad Wessam Alnouri (MPI Bad Nauheim).
Conclusion: The GPCR panel is clean.
| Target protein | HGNC name | Species | RLU [ ] |
|---|---|---|---|
| ADCYAP1R1 | ADCYAP1R1 | Homo sapiens | 1631.2 |
| ADORA1 | ADORA1 | Homo sapiens | 6201.5 |
| ADORA2A | ADORA2A | Homo sapiens | 1002.6 |
| ADORA2B | ADORA2B | Homo sapiens | 6488.0 |
| ADORA3 | ADORA3 | Homo sapiens | 505.9 |
| ADRA1A | ADRA1A | Homo sapiens | 8354.3 |
| ADRA1B | ADRA1B | Homo sapiens | -2728.8 |
| ADRA1D | ADRA1D | Homo sapiens | 2936.5 |
| ADRA2A | ADRA2A | Homo sapiens | 10072.9 |
| ADRA2B | ADRA2B | Homo sapiens | 17935.9 |
| ADRA2C | ADRA2C | Homo sapiens | 12101.9 |
| ADRB1 | ADRB1 | Homo sapiens | 19369.4 |
| ADRB2 | ADRB2 | Homo sapiens | 4582.0 |
| ADRB3 | ADRB3 | Homo sapiens | 12405.3 |
| AGTR1 | AGTR1 | Homo sapiens | 9133.5 |
| AGTR2 | AGTR2 | Homo sapiens | 5320.2 |
| APJ | APLNR | Homo sapiens | 5302.8 |
| AVPR1A | AVPR1A | Homo sapiens | 5668.3 |
| AVPR1B | AVPR1B | Homo sapiens | -688.1 |
| AVPR2 | AVPR2 | Homo sapiens | 2873.6 |
| BB3 | BB3 | Homo sapiens | -2040.2 |
| BDKRB1 | BDKBR1 | Homo sapiens | -3312.8 |
| BDKRB2 | BDKBR2 | Homo sapiens | 892.4 |
| C3AR1 | C3AR1 | Homo sapiens | 4825.0 |
| C5A | C5AR1 | Homo sapiens | 2279.7 |
| CALCRb | CALCR | Homo sapiens | -5810.0 |
| CALCRL | CALCRL | Homo sapiens | 2366.6 |
| CASR | CASR | Homo sapiens | 4396.8 |
| CCKAR | CCKAR | Homo sapiens | 2843.1 |
| CCKBR | CCKBR | Homo sapiens | 2715.7 |
| CCR10 | CCR10 | Homo sapiens | 463.5 |
| CCR2 | CCR2 | Homo sapiens | 2849.0 |
| CCR3 | CCR3 | Homo sapiens | 2423.4 |
| CCR4 | CCR4 | Homo sapiens | 6412.5 |
| CCR5 | CCR5 | Homo sapiens | 2712.2 |
| CCR6 | CCR6 | Homo sapiens | -2062.4 |
| CCR7 | CCR7 | Homo sapiens | 342.3 |
| CCR8 | CCR8 | Homo sapiens | -3273.5 |
| CCRL2 | CCRL2 | Homo sapiens | -1902.1 |
| CD97 | ADGRE5 | Homo sapiens | -894.6 |
| CHRM1 | CHRM1 | Homo sapiens | -2936.3 |
| CHRM2 | CHRM2 | Homo sapiens | -12826.4 |
| CHRM3 | CHRM3 | Homo sapiens | 6260.7 |
| CHRM4 | CHRM4 | Homo sapiens | -837.5 |
| CHRM5 | CHRM5 | Homo sapiens | 7393.2 |
| CMKLR1 | CMKLR1 | Homo sapiens | -332.8 |
| CNR1 | CNR1 | Homo sapiens | -5260.7 |
| CNR2 | CNR2 | Homo sapiens | 4363.5 |
| CRHR1 | CRHR1 | Homo sapiens | 5078.0 |
| CRHR2 | CRHR2 | Homo sapiens | 409.5 |
| CX3C1 | CX3CR1 | Homo sapiens | -3289.6 |
| CXCR1 | CXCR1 | Homo sapiens | 812.1 |
| CXCR2 | CXCR2 | Homo sapiens | -473.1 |
| CXCR3 | CXCR3 | Homo sapiens | -568.0 |
| CXCR4 | CXCR4 | Homo sapiens | -830.7 |
| CXCR5 | CXCR5 | Homo sapiens | -793.2 |
| CXCR6 | CXCR6 | Homo sapiens | 760.7 |
| CXCR7 | ACKR3 | Homo sapiens | -7344.1 |
| CYSLTR1 | CYSLTR1 | Homo sapiens | 1614.6 |
| CYSLTR2 | CYSLTR2 | Homo sapiens | -3192.9 |
| DRD1 | DRD1 | Homo sapiens | 1626.4 |
| DRD2 | DRD2 | Homo sapiens | 2203.4 |
| DRD3 | DRD3 | Homo sapiens | 1163.6 |
| DRD4 | DRD4 | Homo sapiens | -1385.9 |
| DRD5 | DRD5 | Homo sapiens | 856.1 |
| EDNRA | EDNRA | Homo sapiens | -1163.5 |
| EDNRB | EDNRB | Homo sapiens | -88.5 |
| ELTD1 | ADGRL4 | Homo sapiens | 1172.7 |
| F2R | F2R | Homo sapiens | 1351.5 |
| F2RL1 | F2RL1 | Homo sapiens | -1265.2 |
| F2RL2 | F2RL2 | Homo sapiens | 462.8 |
| F2RL3 | F2RL3 | Homo sapiens | 124.5 |
| FFA1 (GPR40) | FFAR1 | Homo sapiens | 2087.7 |
| FFA2 (GPR43) | FFAR2 | Homo sapiens | -5971.4 |
| FFA3 (GPR41) | FFAR3 | Homo sapiens | 1877.4 |
| FPR1 | FPR1 | Homo sapiens | 3268.7 |
| FPR2 | FPR2 | Homo sapiens | 31.8 |
| FPR3 | FPR3 | Homo sapiens | 2837.0 |
| FSHR | FSHR | Homo sapiens | -864.6 |
| G2A | GPR132 | Homo sapiens | -2776.0 |
| GABBR1 | GABBR1 | Homo sapiens | 3394.6 |
| GAL1 | GALR1 | Homo sapiens | -212.4 |
| GAL2 | GALR2 | Homo sapiens | 1135.1 |
| GAL3 | GALR3 | Homo sapiens | -1500.3 |
| GCGR | GCGR | Homo sapiens | 1327.9 |
| GHRHR | GHRHR | Homo sapiens | -1061.4 |
| GHSR | GHSR | Homo sapiens | 1262.8 |
| GIPR | GIPR | Homo sapiens | -1502.2 |
| GLP1R | GLP1R | Homo sapiens | 3482.1 |
| GLP2R | GLP2R | Homo sapiens | -2690.5 |
| GNRHR | GNRHR | Homo sapiens | -3092.9 |
| GPBA | GPBAR1 | Homo sapiens | 275.4 |
| GPER | GPER1 | Homo sapiens | -607.3 |
| GPR1 | GPR1 | Homo sapiens | -60.1 |
| GPR101 | GPR101 | Homo sapiens | -2168.8 |
| GPR110 | ADGRF1 | Homo sapiens | 9363.8 |
| GPR111 | ADGRF2 | Homo sapiens | -1357.3 |
| GPR113 | ADGRF3 | Homo sapiens | 386.5 |
| GPR114 | ADGRG5 | Homo sapiens | 432.5 |
| GPR115 | ADGRF4 | Homo sapiens | -283.1 |
| GPR116 | ADGRF5 | Homo sapiens | -663.5 |
| GPR119 | GPR119 | Homo sapiens | 271.5 |
| GPR12 | GPR12 | Homo sapiens | 109.2 |
| GPR120 | FFAR4 | Homo sapiens | 1034.3 |
| GPR123 | ADGRA1 | Homo sapiens | 2098.3 |
| GPR124 | ADGRA2 | Homo sapiens | -2918.4 |
| GPR125 | ADGRA3 | Homo sapiens | -4100.2 |
| GPR126 | ADGRG6 | Homo sapiens | -6500.1 |
| GPR133 | ADGRD1 | Homo sapiens | -2665.0 |
| GPR135 | GPR135 | Homo sapiens | 2862.2 |
| GPR141 | GPR141 | Homo sapiens | 2790.9 |
| GPR142 | GPR142 | Homo sapiens | 2924.4 |
| GPR143 | GPR143 | Homo sapiens | -2073.8 |
| GPR144 | ADGRD2 | Homo sapiens | 917.4 |
| GPR146 | GPR146 | Homo sapiens | -1507.3 |
| GPR148 | GPR148 | Homo sapiens | 3094.9 |
| GPR149 | GPR149 | Homo sapiens | -2141.6 |
| GPR15 | GPR15 | Homo sapiens | 1711.0 |
| GPR150 | GPR150 | Homo sapiens | -1602.2 |
| GPR151 | GPR151 | Homo sapiens | 12913.8 |
| GPR152 | GPR152 | Homo sapiens | -70.0 |
| GPR153 | GPR153 | Homo sapiens | -4686.9 |
| GPR156 | GPR156 | Homo sapiens | 1544.4 |
| GPR157 | GPR157 | Homo sapiens | -4179.8 |
| GPR158 | GPR158 | Homo sapiens | 1540.2 |
| GPR160 | GPR160 | Homo sapiens | 1902.7 |
| GPR161 | GPR161 | Homo sapiens | -2638.3 |
| GPR162 | GPR162 | Homo sapiens | 6270.0 |
| GPR17 | GPR17 | Homo sapiens | 896.7 |
| GPR171 | GPR171 | Homo sapiens | -3245.4 |
| GPR173 | GPR173 | Homo sapiens | -36.4 |
| GPR174 | GPR174 | Homo sapiens | -102.0 |
| GPR18 | GPR18 | Homo sapiens | -382.9 |
| GPR182 | GPR182 | Homo sapiens | 598.2 |
| GPR183 | GPR183 | Homo sapiens | -6103.2 |
| GPR19 | GPR19 | Homo sapiens | 1532.0 |
| GPR20 | GPR20 | Homo sapiens | -1202.2 |
| GPR21 | GPR21 | Homo sapiens | -483.4 |
| GPR22 | GPR22 | Homo sapiens | -1209.1 |
| GPR25 | GPR25 | Homo sapiens | -1214.2 |
| GPR26 | GPR26 | Homo sapiens | -186.7 |
| GPR27 | GPR27 | Homo sapiens | -2082.3 |
| GPR3 | GPR3 | Homo sapiens | -1785.0 |
| GPR31 | GPR31 | Homo sapiens | 1301.8 |
| GPR32 | GPR32 | Homo sapiens | 5658.8 |
| GPR34 | GPR34 | Homo sapiens | 5570.9 |
| GPR35 | GPR35 | Homo sapiens | 2600.5 |
| GPR37 | GPR37 | Homo sapiens | -1507.2 |
| GPR37L1 | GPR37L1 | Homo sapiens | 152895.5 |
| GPR39 | GPR39 | Homo sapiens | 8022.0 |
| GPR4 | GPR4 | Homo sapiens | -970.1 |
| GPR44 | PTGDR2 | Homo sapiens | -285.1 |
| GPR45 | GPR45 | Homo sapiens | 963.5 |
| GPR50 | GPR50 | Homo sapiens | 435058.5 |
| GPR52 | GPR52 | Homo sapiens | 86517.0 |
| GPR55 | GPR55 | Homo sapiens | 601993.4 |
| GPR56 | ADGRG1 | Homo sapiens | 14078.3 |
| GPR6 | GPR6 | Homo sapiens | 1071405.4 |
| GPR61 | GPR61 | Homo sapiens | 1404.9 |
| GPR62 | GPR62 | Homo sapiens | 477269.9 |
| GPR63 | GPR63 | Homo sapiens | -87.9 |
| GPR64 | ADGRG2 | Homo sapiens | 8730.8 |
| GPR65 | GPR65 | Homo sapiens | -1353.6 |
| GPR68 | GPR68 | Homo sapiens | -1793.0 |
| GPR75 | GPR75 | Homo sapiens | 867.6 |
| GPR77 | C5AR2 | Homo sapiens | 350.6 |
| GPR78 | GPR78 | Homo sapiens | 5.4 |
| GPR82 | GPR82 | Homo sapiens | -8045.7 |
| GPR83 | GPR83 | Homo sapiens | 834.2 |
| GPR84 | GPR84 | Homo sapiens | -3986.6 |
| GPR85 | GPR85 | Homo sapiens | -4210.7 |
| GPR87 | GPR87 | Homo sapiens | 8749.9 |
| GPR88 | GPR88 | Homo sapiens | 162.4 |
| GPR97 | ADGRG3 | Homo sapiens | 2049.6 |
| GPRC5A | GPRC5A | Homo sapiens | 3572.6 |
| GPRC5B | GPRC5B | Homo sapiens | -3638.3 |
| GPRC5C | GPRC5C | Homo sapiens | 3557.1 |
| GPRC5D | GPRC5D | Homo sapiens | 1.7 |
| GPRC6A | GPRC6A | Homo sapiens | -9108.7 |
| GRM1 | GRM1 | Homo sapiens | -510.5 |
| GRM2 | GRM2 | Homo sapiens | -1461.8 |
| GRM4 | GRM4 | Homo sapiens | -82.8 |
| GRM5 | GRM5 | Homo sapiens | -10050.2 |
| GRM6 | GRM6 | Homo sapiens | -158.4 |
| GRM7 | GRM7 | Homo sapiens | 6954.3 |
| GRM8 | GRM8 | Homo sapiens | -4064.9 |
| GRPR | GRPR | Homo sapiens | -1247.8 |
| HCA1 | HCAR1 | Homo sapiens | 582.5 |
| HCA2 | HCAR2 | Homo sapiens | -133.2 |
| HCA3 | HCAR3 | Homo sapiens | 1810.9 |
| HCTR1 | SLC31A1 | Homo sapiens | -2836.0 |
| HCTR2 | SLC31A2 | Homo sapiens | 2837.4 |
| HRH1 | HRH1 | Homo sapiens | 13456.2 |
| HRH2 | HRH2 | Homo sapiens | 84.8 |
| HRH3 | HRH3 | Homo sapiens | -6781.6 |
| HRH4 | HRH4 | Homo sapiens | -637.3 |
| HTR1A | HTR1A | Homo sapiens | 1526.2 |
| HTR1B | HTR1B | Homo sapiens | 77.2 |
| HTR1D | HTR1D | Homo sapiens | -12275.7 |
| HTR1E | HTR1E | Homo sapiens | -637.5 |
| HTR1F | HTR1F | Homo sapiens | -3470.8 |
| HTR2A | HTR2A | Homo sapiens | -2874.2 |
| HTR2B | HTR2B | Homo sapiens | -1737.0 |
| HTR2C | HTR2C | Homo sapiens | 1050.5 |
| HTR4 | HTR4 | Homo sapiens | -2332.3 |
| HTR5 | HTR5 | Homo sapiens | -1883.4 |
| HTR6 | HTR6 | Homo sapiens | 5341.3 |
| HTR7 | HTR7 | Homo sapiens | -1000.9 |
| KISSPEPTIN | KISS1R | Homo sapiens | 2036.6 |
| LHCGR | LHCGR | Homo sapiens | 153.9 |
| LPAR1 | LPAR1 | Homo sapiens | 280.0 |
| LPAR2 | LPAR2 | Homo sapiens | -80.0 |
| LPAR4 | LPAR4 | Homo sapiens | -668.3 |
| LPAR5 | LPAR5 | Homo sapiens | 471.2 |
| LPAR6 | LPAR6 | Homo sapiens | -7371.4 |
| LTB4R | LTB4R | Homo sapiens | -269.9 |
| LTB4R2B | LTB4R2 | Homo sapiens | 300919.8 |
| MAS1 | MAS1 | Homo sapiens | -1359.6 |
| MAS1L | MAS1L | Homo sapiens | 2608.3 |
| MC1R | MC1R | Homo sapiens | -1886.9 |
| MC2R | MC2R | Homo sapiens | 1069.0 |
| MC3R | MC3R | Homo sapiens | 18.8 |
| MC4R | MC4R | Homo sapiens | -2107.5 |
| MC5R | MC5R | Homo sapiens | 481.1 |
| MCHR1 | MCHR1 | Homo sapiens | 5932.9 |
| MCHR2 | MCHR2 | Homo sapiens | 1.7 |
| MLNR | MLNR | Homo sapiens | -569.6 |
| MRGPRD | MRGPRD | Homo sapiens | -630.4 |
| MRGPRE | MRGPRE | Homo sapiens | -3205.5 |
| MRGPRF | MRGPRF | Homo sapiens | -194.1 |
| MRGPRG | MRGPRG | Homo sapiens | -559.7 |
| MRGPRX1 | MRGPRX1 | Homo sapiens | 319.1 |
| MRGPRX2 | MRGPRX2 | Homo sapiens | -9422.3 |
| MRGPRX3 | MRGPRX3 | Homo sapiens | -915.6 |
| MRGPRX4 | MRGPRX4 | Homo sapiens | 3306.4 |
| MTNR1A | MTNR1A | Homo sapiens | 466.4 |
| MTNR1B | MTNR1B | Homo sapiens | 4173.8 |
| NMBR | NMBR | Homo sapiens | 937.3 |
| NMUR1 | NMUR1 | Homo sapiens | 1954.2 |
| NMUR2 | NMUR2 | Homo sapiens | 710.0 |
| NPBW1 | NPBWR1 | Homo sapiens | 4937.6 |
| NPBW2 | NPBWR2 | Homo sapiens | -872.1 |
| NPFF1 | NPFFR1 | Homo sapiens | 4030.1 |
| NPFF2 | NPFFR2 | Homo sapiens | -116.2 |
| NPS | NPSR1 | Homo sapiens | 3786.6 |
| NPY1R | NPY1R | Homo sapiens | -114.3 |
| NPY2R | NPY2R | Homo sapiens | 558.7 |
| NPY4R | NPY4R | Homo sapiens | -158.1 |
| NPY5R | NPY5R | Homo sapiens | -14453.5 |
| NTSR1 | NTSR1 | Homo sapiens | -1298.1 |
| NTSR2 | NTSR2 | Homo sapiens | 633.7 |
| OPN3 | OPN3 | Homo sapiens | 338.2 |
| OPN5 | OPN5 | Homo sapiens | 3998.2 |
| OPRD1 | OPRD1 | Homo sapiens | 1287.2 |
| OPRK1 | OPRK1 | Homo sapiens | 156.1 |
| OPRL1 | OPRL1 | Homo sapiens | 2755.3 |
| OPRM1 | OPRM1 | Homo sapiens | 3974.9 |
| OXER1 | OXER1 | Homo sapiens | -152.7 |
| OXGR1 | OXGR1 | Homo sapiens | -825.6 |
| OXTR | OXTR | Homo sapiens | -478.7 |
| P2RY1 | P2RY1 | Homo sapiens | 1691.9 |
| P2RY10 | P2RY10 | Homo sapiens | -82.4 |
| P2RY11 | P2RY11 | Homo sapiens | -216.0 |
| P2RY12 | P2RY12 | Homo sapiens | -34.3 |
| P2RY13 | P2RY13 | Homo sapiens | 10145.0 |
| P2RY14 | P2RY14 | Homo sapiens | -5257.2 |
| P2RY2 | P2RY2 | Homo sapiens | 2247.4 |
| P2RY4 | P2RY4 | Homo sapiens | -311.1 |
| P2RY6 | P2RY6 | Homo sapiens | -7244.2 |
| P2RY8 | P2RY8 | Homo sapiens | 1325.5 |
| PK1 | PROKR1 | Homo sapiens | 10848.1 |
| PK2 | PROKR2 | Homo sapiens | -566.0 |
| PRRP | PRLHR | Homo sapiens | 4140.2 |
| PTAFR | PTAFR | Homo sapiens | 82.9 |
| PTGDR | PTGDR | Homo sapiens | 375.1 |
| PTGER1 | PTGER1 | Homo sapiens | -390.2 |
| PTGER2 | PTGER2 | Homo sapiens | 612.9 |
| PTGER3 | PTGER3 | Homo sapiens | 83.2 |
| PTGER4 | PTGER4 | Homo sapiens | 620.1 |
| PTGFR | PTGFR | Homo sapiens | -81.2 |
| PTGIR | PTGIR | Homo sapiens | -407.6 |
| PTH1R | PTH1R | Homo sapiens | 13.4 |
| PTH2R | PTH2R | Homo sapiens | -1532.5 |
| QRFP | QRFP | Homo sapiens | -576.6 |
| RXFP1 | RXFP1 | Homo sapiens | -1130.3 |
| RXFP2 | RXFP2 | Homo sapiens | -899.8 |
| RXFP3 | RXFP3 | Homo sapiens | 6608.6 |
| RXFP4 | RXFP4 | Homo sapiens | 68.6 |
| S1PR1 | S1PR1 | Homo sapiens | 11032.9 |
| S1PR2 | S1PR2 | Homo sapiens | 401.1 |
| S1PR3 | S1PR3 | Homo sapiens | -1651.7 |
| S1PR4 | S1PR4 | Homo sapiens | -471.1 |
| S1PR5 | S1PR5 | Homo sapiens | 2920.1 |
| SCTR | SCTR | Homo sapiens | -71.4 |
| SSTR1 | SSTR1 | Homo sapiens | -1071.3 |
| SSTR2 | SSTR2 | Homo sapiens | -162.6 |
| SSTR3 | SSTR3 | Homo sapiens | 342.4 |
| SSTR4 | SSTR4 | Homo sapiens | 120.1 |
| SSTR5 | SSTR5 | Homo sapiens | -945.6 |
| SUCNR1 | SUCNR1 | Homo sapiens | 1538.4 |
| TA1 | TAAR1 | Homo sapiens | 127.2 |
| TAAR2 | TAAR2 | Homo sapiens | 390.1 |
| TAAR5 | TAAR5 | Homo sapiens | 821.2 |
| TAAR6 | TAAR6 | Homo sapiens | -393.5 |
| TAAR8 | TAAR8 | Homo sapiens | -4861.1 |
| TAAR9 | TAAR9 | Homo sapiens | -546.9 |
| TACR1 | TACR1 | Homo sapiens | -4718.2 |
| TACR2 | TACR2 | Homo sapiens | -238.0 |
| TACR3 | TACR3 | Homo sapiens | 549.7 |
| TBXA2R | TBXA2R | Homo sapiens | 232.6 |
| TSHR | TSHR | Homo sapiens | -405.9 |
| UTS2R | UTS2R | Homo sapiens | -160.1 |
| VIPR1 | VIPR1 | Homo sapiens | -7193.3 |
| VIPR2 | VIPR2 | Homo sapiens | -823.8 |