Physicochemical properties of probe BI-8668 and control BI-0337
| BI-8668 | |
|---|---|
| log D (pH 7.4) | 0.2 |
| log D (pH 2) | -0.5 |
| log D (pH 11) | 0.6 |
| BI-0337 | |
|---|---|
| log D (pH 2) | -0.8 |
Solubility
| BI-8668: |
PBS pH 7.4: 110 µg/mL
|
| BI-0337: |
PBS pH 7.4: 81 µg/mL
|
| BI-8668 | |
|---|---|
| log D (pH 7.4) | 0.2 |
| log D (pH 2) | -0.5 |
| log D (pH 11) | 0.6 |
| BI-0337 | |
|---|---|
| log D (pH 2) | -0.8 |
| BI-8668: |
PBS pH 7.4: 110 µg/mL
|
| BI-0337: |
PBS pH 7.4: 81 µg/mL
|