Physicochemical properties of GSK973
| GSK973 | |
|---|---|
| Artificial Membrane Permeability (AMP) | 165 nM/s |
| Appearance | colorless solid |
| Chrom log D pH 7.4 | 3.6 |
Solubility
| GSK973: |
Kinetic aqueous solubility measured with Chemiluminescent Nitrogen Detection (CLND): 173 µg/mL, 
FaSSIF (fasted state simulated intestinal fluid): 80 µg/mL
|