Potency data for probe BI 665915 and control BI-0153
In vitro potency
| Target name | Target information | Species | Assay description | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|
| ALOX5AP | Homo sapiens | Binding assay: Geometric mean values (n >= 3), each determined from duplicate 10-point concentration-response curves. | IC50 = 1.700 nM | IC50 = 670 nM |
In cell potency
| Target name | Target information | Species | Assay description | Probe result (SD) | Control result (SD) | Publication of assay conditions |
|---|---|---|---|---|---|---|
| ALOX5AP | Homo sapiens | Functional inhibition in human whole blood: Geometric mean values (n >= 3), each determined from duplicate 10-point concentration-response curves. | IC50 = 45 nM | |||
| ALOX5AP | Mus musculus | Functional inhibition in mouse whole blood: Geometric mean values (n >= 3), each determined from duplicate 8-point concentration-response curves. | IC50 = 4800 nM |