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Selectivity data for probe TP-030-1 and control TP-030n


Jump to control PDSP data

TP-030-1


Compound concentration: 10 µM
Receptor HGNC target name Inhibition [%] (Primary experimental value) Ki [nM] (Secondary experimental value) pKi
Beta1 ADRB1 5.21
Beta3 ADRB3 9.80
GABAA/BZP -3.98
GABAA 10.49
GABA/PBR 68.73 374.92 average (n=2) 6.43
D4 DRD4 17.41
D5 DRD5 1.77
DAT SLC6A3 -11.53
H4 HRH4 6.09
KOR OPRK1 14.71
MOR OPRM1 10.56
Alpha1A ADRA1A -0.50
Alpha1B ADRA1B -13.41
Alpha1D ADRA1D -0.30
Alpha2A ADRA2A 19.06
Alpha2B ADRA2B 43.34
Alpha2C ADRA2C 34.69
M1 CHRM1 0.60
M2 CHRM2 -4.37
M3 CHRM3 0.09
M5 CHRM5 6.63
Sigma 1 SIGMAR1 -1.90
Sigma 2 TMEM97 27.01
5-HT1A HTR1A 5.07
5-HT1B HTR1B 0.99
5-HT1D HTR1D -13.67
5-HT1E HTR1E -1.55
5-HT2A HTR2A 3.80
5-HT2B HTR2B 12.00
5-HT6 HTR6 -3.95
5-HT7A HTR7 -1.17
D1 DRD1 18.79
D2 DRD2 -5.46
D3 DRD3 -4.81
5-HT2C HTR2C -2.89
5-HT3 HTR3A 40.83
5-HT5A HTR5A 21.09
Beta2 ADRB2 9.59
DOR OPRD1 28.83
H1 HRH1 20.53
H2 HRH2 11.93
H3 HRH3 -19.63
M4 CHRM4 8.56
NET SLC6A2 -12.17
SERT SLC6A4 5.99

Jump to PDSP top

TP-030-1

Results are significant for > 50 % inhibition. Where presented, IC50 values were determined by a non-linear, least squares regression analysis using MathIQTM (ID Business Solutions Ltd., UK). The inhibition constants (Ki) were calculated with the equation of Cheng and Prusoff (Cheng, Y., Prusoff, W.H., Biochem. Pharmacol. 22:3099-3108, 1973) using the observed IC50 value of the tested compound, the concentration of radioligand employed in the assay, and the historical values for the Ki of the ligand (obtained experimentally at MDS Pharma Services).

Conclusion: Clean panel.

Target protein HGNC name Species Cmp. conc. % inhibition Reference compound name Reference compound IC50 [nM] Assay ID
Adenosine A1 ADORA1 Homo sapiens 10 µM 7.0 R(-)-PIA 830.00 200510
Adenosine A2A ADORA2A Homo sapiens 10 µM 10.0 CGS-Z1680 130.00 200610
Adenosine A3 ADORA3 Homo sapiens 10 µM 15.0 IB-MECA 0.78 200720
Adrenergic alpha1A ADRA1A Homo sapiens 10 µM -1.0 Prazosin hydrochloride 0.87 203110
Adrenergic alpha1B ADRA1B Homo sapiens 10 µM 2.0 Prazosin hydrochloride 0.25 203210
Adrenergic alpha1D ADRA1D Homo sapiens 10 µM -2.0 Prazosin 0.88 203400
Adrenergic alpha2A ADRA2A Homo sapiens 10 µM 7.0 Yohimbine 1.80 203630
Adrenergic beta1 ADRB1 Homo sapiens 10 µM -8.0 S(-)-Propranolol 2.50 204010
Adrenergic beta2 ADRB2 Homo sapiens 10 µM -4.0 S(-)-Propranolol 0.78 204110
Androgen (Testosterone) AR AR Homo sapiens 10 µM 6.0 Testosterone 2.10 206000
Bradykinin B1 BDKRB1 Homo sapiens 10 µM 2.0 (Des-Arg10)-Kallidin 0.29 212520
Bradykinin B2 BDKRB2 Homo sapiens 10 µM 4.0 Bradykinin 1.80 212620
Calcium Channel L-Type, Benzothiazepine CACNA1C Rattus sp. 10 µM 23.0 Diltiazem 0.04 214510
Calcium Channel L-Type, Dihydropyridine CACNA1C Rattus sp. 10 µM -18.0 Nitrendipine 0.72 214600
Calcium Channel N-Type CACNA1B Rattus sp. 10 µM -2.0 omega-Conotoxin GVIA 0.03 216000
Cannabinoid CB1 CNR1 Homo sapiens 10 µM 5.0 CP-55,940 33.00 217050
Dopamine D1 DRD1 Homo sapiens 10 µM -4.0 R(+)-SCH-Z3390 1.40 219500
Dopamine D2S DRD2 Homo sapiens 10 µM 7.0 Spiperone 0.25 219700
Dopamine D3 DRD3 Homo sapiens 10 µM 8.0 Spiperone 0.36 219800
Dopamine D4.4 DRD5 Homo sapiens 10 µM 3.0 Spiperone 0.76 220200
Endothelin ETA EDNRA Homo sapiens 10 µM -5.0 Endothelin-1 0.23 224010
Endothelin ETB EDNRB Homo sapiens 10 µM 0.0 Endothelin-1 0.13 224110
Epidermal Growth Factor (EGF) EGFR Homo sapiens 10 µM -3.0 EGF (human) 1.60 225510
Estrogen ERalpha ESR1 Homo sapiens 10 µM 36.0 Diethylstilbestrol 0.77 226010
GABAA, Flunitrazepam, Central Rattus sp. 10 µM 8.0 Hydrogen diazepam chloride 16.00 226600
GABAA, Muscimol, Central Rattus sp. 10 µM -1.0 GABA 32.00 226500
GABAB1A GABBR1 Homo sapiens 10 µM 0.0 Cgp-54626 6.40 228610
Glucocorticoid NR3C1 Homo sapiens 10 µM 5.0 Dexamethasone 3.80 232030
Glutamate, Kainate Rattus sp. 10 µM -2.0 L-Glutamic acid hydrochloride 160.00 232710
Glutamate, NMDA, Agonism Rattus sp. 10 µM -13.0 L-Glutamic acid 410.00 232810
Glutamate, NMDA, Glycine Rattus sp. 10 µM 0.0 MDL 105,519 22.00 232910
Glutamate, NMDA, Phencyclidine Rattus sp. 10 µM -8.0 Dizolcipine ((+)-MK-801) 5.10 233000
Histamine H1 HRH1 Homo sapiens 10 µM 3.0 Pyrilamine 3.30 239610
Histamine H2 HRH2 Homo sapiens 10 µM -12.0 Tiotidine 22.00 239710
Histamine H3 HRH3 Homo sapiens 10 µM 4.0 R(-)-alpha-Methylhistamine (RAMH) 2.30 239820
Imidazoline I2, Central Rattus sp. 10 µM 6.0 Idazoxan 12.00 241000
Interleukin IL-1 R1 IL1R1 Homo sapiens 10 µM -7.0 IL-1 beta 1.80 243530
Leukotriene, Cysteinyl CysLT1 CYSLTR1 Homo sapiens 10 µM 0.0 Leukotriene D4 0.70 250460
Melatonin MT1 MTNR1A Homo sapiens 10 µM 45.0 Melatonin 0.21 251600
Muscarinic M1 CHRM1 Homo sapiens 10 µM 0.0 4-DAMP 4.50 252610
Muscarinic M2 CHRM2 Homo sapiens 10 µM -4.0 4-DAMP 55.00 252710
Muscarinic M3 CHRM3 Homo sapiens 10 µM 1.0 4-DAMP 5.10 252810
Neuropeptide Y Y1 NPY1R Homo sapiens 10 µM 4.0 Neuropeptide Y (human, rat) 0.22 257010
Neuropeptide Y Y2 NPY2R Homo sapiens 10 µM 2.0 Neuropeptide Y (13-36) (porcine) 0.21 257110
Nicotinic Acetylcholine alpha1, Bungarotoxin CHRNA1 Homo sapiens 10 µM -8.0 alpha-Bungarotoxin 1.10 258700
Nicotinic Acetylcholine alpha3beta4 CHRNA3
CHRNB4
Homo sapiens 10 µM 21.0 (-)-Epibatidine 0.10 258730
Opiate delta1 (OP1, DOP) OPRD1 Homo sapiens 10 µM 3.0 Naltrindole 0.91 260130
Opiate kappa (OP2, KOP) OPRK1 Homo sapiens 10 µM 3.0 U-69593 16.00 260210
Opiate µ (OP3, MOP) OPRM1 Homo sapiens 10 µM 19.0 DAMGO 20.00 260410
Phorbol Ester Mus musculus 10 µM -3.0 Phorbol myristate acetate 0.79 264500
Platelet Activating Factor (PAF) PTAFR Homo sapiens 10 µM 2.0 PAF 1.80 299037
Potassium Channel [KATP] KCNJ11 Cricetinae 10 µM 6.0 Glyburide 5.70 265600
Potassium Channel hERG KCNH2 Homo sapiens 10 µM -5.0 Astemizole 2.60 265900
Prostanoid EP4 PTGER4 Homo sapiens 10 µM 12.0 Prostaglandin E2 (PGE2) 1.10 268420
Purinergic P2X Rattus sp. 10 µM -6.0 Alpha, beta-Methylene ATP 11.00 299036
Purinergic P2Y Rattus sp. 10 µM -5.0 2-Methylthio-ATP 85.00 268820
Rolipram Rattus sp. 10 µM 0.0 Rolipram 5.70 270000
Serotonin (5-Hydroxytryptamine) 5-HT1A HTR1A Homo sapiens 10 µM -6.0 Metergoline 4.10 271110
Serotonin (5-Hydroxytryptamine) 5-HT2B HTR2B Homo sapiens 10 µM 6.0 Ketanserin 290.00 271700
Serotonin (5-Hydroxytryptamine) 5-HT3 HTR3A Homo sapiens 10 µM 6.0 MDL-72222 11.00 271910
Sigma 1 SIGMAR1 Homo sapiens 10 µM 27.0 Haloperidol 6.42 299034
Sodium Channel, Site 2 Rattus sp. 10 µM 46.0 Dibucaine 61.00 279510
Tachykinin NK1 TACR1 Homo sapiens 10 µM 29.0 L-703606 3.60 255520
Thyroid Hormone Rattus sp. 10 µM 24.0 Liothyronine 0.03 285900
Transporter, Dopamine (DAT) SLC6A3 Homo sapiens 10 µM 29.0 GBR-12909 1.70 220320
Transporter, GABA Rattus sp. 10 µM -7.0 NO-711 200.00 226400
Transporter, Norepinephrine (NET) SLC6A2 Homo sapiens 10 µM 15.0 Desipramine 0.93 204410
Transporter, Serotonin (5- Hydroxytryptamine) (SERT) SLC6A4 Homo sapiens 10 µM -4.0 Fluoxetine 8.60 274030
 

TP-030n

Conclusion: Clean panel.

Target protein HGNC name Species Cmp. conc. % inhibition Reference compound name Reference compound IC50 [nM] Assay ID
Adenosine A1 ADORA1 Homo sapiens 10 µM -2.0 R(-)-PIA 830.0 200510
Adenosine A2A ADORA2A Homo sapiens 10 µM -8.0 CGS-Z1680 130.0 200610
Adenosine A3 ADORA3 Homo sapiens 10 µM -33.0 IB-MECA 0.8 200720
Adrenergic alpha1A ADRA1A Homo sapiens 10 µM 1.0 Prazosin hydrochloride 0.9 203110
Adrenergic alpha1B ADRA1B Homo sapiens 10 µM 1.0 Prazosin hydrochloride 0.3 203210
Adrenergic alpha1D ADRA1D Homo sapiens 10 µM -19.0 Prazosin 0.9 203400
Adrenergic alpha2A ADRA2A Homo sapiens 10 µM -16.0 Yohimbine 1.8 203630
Adrenergic beta1 ADRB1 Homo sapiens 10 µM -12.0 S(-)-Propranolol 2.5 204010
Adrenergic beta2 ADRB2 Homo sapiens 10 µM 4.0 S(-)-Propranolol 0.8 204110
Androgen (Testosterone) AR AR Homo sapiens 10 µM 0.0 Testosterone 2.1 206000
Bradykinin B1 BDKRB1 Homo sapiens 10 µM 9.0 (Des-Arg10)-Kallidin 0.3 212520
Bradykinin B2 BDKRB2 Homo sapiens 10 µM -4.0 Bradykinin 1.8 212620
Calcium Channel L-Type, Benzothiazepine CACNA1C Rattus sp. 10 µM 2.0 Diltiazem 0.0 214510
Calcium Channel L-Type, Dihydropyridine CACNA1C Rattus sp. 10 µM -6.0 Nitrendipine 0.7 214600
Calcium Channel N-Type CACNA1B Rattus sp. 10 µM 2.0 omega-Conotoxin GVIA 0.0 216000
Cannabinoid CB1 CNR1 Homo sapiens 10 µM -5.0 CP-55,940 33.0 217050
Dopamine D1 DRD1 Homo sapiens 10 µM 7.0 R(+)-SCH-Z3390 1.4 219500
Dopamine D2S DRD2 Homo sapiens 10 µM 2.0 Spiperone 0.3 219700
Dopamine D3 DRD3 Homo sapiens 10 µM 4.0 Spiperone 0.4 219800
Dopamine D4.4 DRD5 Homo sapiens 10 µM 3.0 Spiperone 0.8 220200
Endothelin ETA EDNRA Homo sapiens 10 µM -12.0 Endothelin-1 0.2 224010
Endothelin ETB EDNRB Homo sapiens 10 µM -3.0 Endothelin-1 0.1 224110
Epidermal Growth Factor (EGF) EGFR Homo sapiens 10 µM 4.0 EGF (human) 1.6 225510
Estrogen ERalpha ESR1 Homo sapiens 10 µM 5.0 Diethylstilbestrol 0.8 226010
GABAA, Flunitrazepam, Central Rattus sp. 10 µM 12.0 Hydrogen diazepam chloride 16.0 226600
GABAA, Muscimol, Central Rattus sp. 10 µM -7.0 GABA 32.0 226500
GABAB1A GABBR1 Homo sapiens 10 µM -6.0 Cgp-54626 6.4 228610
Glucocorticoid NR3C1 Homo sapiens 10 µM 3.0 Dexamethasone 3.8 232030
Glutamate, Kainate Rattus sp. 10 µM 7.0 L-Glutamic acid hydrochloride 160.0 232710
Glutamate, NMDA, Agonism Rattus sp. 10 µM 4.0 L-Glutamic acid 410.0 232810
Glutamate, NMDA, Glycine Rattus sp. 10 µM -2.0 MDL 105,519 22.0 232910
Glutamate, NMDA, Phencyclidine Rattus sp. 10 µM -9.0 Dizolcipine ((+)-MK-801) 5.1 233000
Histamine H1 HRH1 Homo sapiens 10 µM 8.0 Pyrilamine 3.3 239610
Histamine H2 HRH2 Homo sapiens 10 µM -10.0 Tiotidine 22.0 239710
Histamine H3 HRH3 Homo sapiens 10 µM -5.0 R(-)-alpha-Methylhistamine (RAMH) 2.3 239820
Imidazoline I2, Central Rattus sp. 10 µM -28.0 Idazoxan 12.0 241000
Interleukin IL-1 R1 IL1R1 Homo sapiens 10 µM -9.0 IL-1 beta 1.8 243530
Leukotriene, Cysteinyl CysLT1 CYSLTR1 Homo sapiens 10 µM 0.0 Leukotriene D4 0.7 250460
Melatonin MT1 MTNR1A Homo sapiens 10 µM 9.0 Melatonin 0.2 251600
Muscarinic M1 CHRM1 Homo sapiens 10 µM 2.0 4-DAMP 4.5 252610
Muscarinic M2 CHRM2 Homo sapiens 10 µM 9.0 4-DAMP 55.0 252710
Muscarinic M3 CHRM3 Homo sapiens 10 µM -3.0 4-DAMP 5.1 252810
Neuropeptide Y Y1 NPY1R Homo sapiens 10 µM -3.0 Neuropeptide Y (human, rat) 0.2 257010
Neuropeptide Y Y2 NPY2R Homo sapiens 10 µM 1.0 Neuropeptide Y (13-36) (porcine) 0.2 257110
Nicotinic Acetylcholine alpha1, Bungarotoxin CHRNA1 Homo sapiens 10 µM -13.0 alpha-Bungarotoxin 1.1 258700
Nicotinic Acetylcholine alpha3beta4 CHRNA3
CHRNB4
Homo sapiens 10 µM 2.0 (-)-Epibatidine 0.1 258730
Opiate delta1 (OP1, DOP) OPRD1 Homo sapiens 10 µM -8.0 Naltrindole 0.9 260130
Opiate kappa (OP2, KOP) OPRK1 Homo sapiens 10 µM 3.0 U-69593 16.0 260210
Opiate µ (OP3, MOP) OPRM1 Homo sapiens 10 µM 4.0 DAMGO 20.0 260410
Phorbol Ester Mus musculus 10 µM 7.0 Phorbol myristate acetate 0.8 264500
Platelet Activating Factor (PAF) PTAFR Homo sapiens 10 µM -24.0 PAF 1.8 299037
Potassium Channel [KATP] KCNJ11 Cricetinae 10 µM 5.0 Glyburide 5.7 265600
Potassium Channel hERG KCNH2 Homo sapiens 10 µM 11.0 Astemizole 2.6 265900
Prostanoid EP4 PTGER4 Homo sapiens 10 µM -19.0 Prostaglandin E2 (PGE2) 1.1 268420
Purinergic P2X Rattus sp. 10 µM -19.0 Alpha, beta-Methylene ATP 11.0 299036
Purinergic P2Y Rattus sp. 10 µM 8.0 2-Methylthio-ATP 85.0 268820
Rolipram Rattus sp. 10 µM 1.0 Rolipram 5.7 270000
Serotonin (5-Hydroxytryptamine) 5-HT1A HTR1A Homo sapiens 10 µM 3.0 Metergoline 4.1 271110
Serotonin (5-Hydroxytryptamine) 5-HT2B HTR2B Homo sapiens 10 µM -2.0 Ketanserin 290.0 271700
Serotonin (5-Hydroxytryptamine) 5-HT3 HTR3A Homo sapiens 10 µM 16.0 MDL-72222 11.0 271910
Sigma 1 SIGMAR1 Homo sapiens 10 µM 11.0 Haloperidol 6.4 299034
Sodium Channel, Site 2 Rattus sp. 10 µM 9.0 Dibucaine 61.0 279510
Tachykinin NK1 TACR1 Homo sapiens 10 µM 14.0 L-703606 3.6 255520
Thyroid Hormone Rattus sp. 10 µM 21.0 Liothyronine 0.0 285900
Transporter, Dopamine (DAT) SLC6A3 Homo sapiens 10 µM 10.0 GBR-12909 1.7 220320
Transporter, GABA Rattus sp. 10 µM -11.0 NO-711 200.0 226400
Transporter, Norepinephrine (NET) SLC6A2 Homo sapiens 10 µM 3.0 Desipramine 0.9 204410
Transporter, Serotonin (5- Hydroxytryptamine) (SERT) SLC6A4 Homo sapiens 10 µM 5.0 Fluoxetine 8.6 274030

TP-030-1

For this kinase screen a competitive binding assay with a fluorescent probe compound was used as decribed in Hirozane et al.. The kinase panel assay was performed at 1000 nM and 100 nM. pIC50 values were calculated by fitting the data to a sigmoidal dose response curve with fixed parameters, top = 100% inhibition, bottom = 0% inhibition and hill slope =1, using XLfit software developed by IDBS. pIC50 cut off value = 6.0.

Conclusion: Clean panel. Only hit is the target RIPK1 of the inhibitor with pIC50 = 7.66.

Target protein HGNC name Species pIC50
Abl(ABL1IHY1) ABL1 Homo sapiens 6.0
Arg(ABL2LGF1) ABL2 Homo sapiens 6.0
ALK2(ACV1LGF1) ACVR1 Homo sapiens 6.0
ACtR2(AC2ALGE1) ACVR2A Homo sapiens 6.0
ALK1(ACL1LGF1) ACVRL1 Homo sapiens 6.0
BARK1 [GRK2(ADR1LGG5)] GRK2 Homo sapiens 6.0
BARK2 [GRK3(ADR2LGG5)] GRK3 Homo sapiens 6.0
Akt2 [PKBbeta(AKT2CGY1)] AKT2 Homo sapiens 6.0
Akt3 [PKBgamma(AKT3LGY1)] AKT3 Homo sapiens 6.0
ALK(ALK1LGY1) ALK Homo sapiens 6.0
SgK288(ANK1LGRL) ANKK1 Homo sapiens 6.0
AurA [Aur2(AURALGF1)] AURKA Homo sapiens 6.0
AurB [Aur1(AURBPGE1)] AURKB Homo sapiens 6.0
Axl(AXL1LGY1) AXL Homo sapiens 6.0
BLK(BLK1CGF1) BLK Homo sapiens 6.0
BIKE(BM2KLGY1) BMP2K Homo sapiens 6.0
BMPR1A(BM1APHRG) BMPR1A Homo sapiens 6.0
BMPR1B(BM1BLGF1) BMPR1B Homo sapiens 6.0
BMPR2(BMR2LGN1) BMPR2 Homo sapiens 6.0
Etk [BMX(BMX1CGF1)] BMX Homo sapiens 6.0
BRAF(BRAFLGY1) BRAF Homo sapiens 6.0
BRSK1(BRS1LGA1) BRSK1 Homo sapiens 6.0
BTK(BTK1CGF1) BTK Homo sapiens 6.0
Bub1(BUB1LGRL) BUB1 Homo sapiens 6.0
CaMK1gamma(CA1GLGN1) CAMK1G Homo sapiens 6.0
CaMK4(CAM4LGY1) CAMK4 Homo sapiens 6.0
CASK(CASKLGY1) CASK Homo sapiens 6.0
MRCKalpha(CD4ALGY1) CDC42BPA Homo sapiens 6.0
DMPK2(CD4GLGRD) EPHB1 Homo sapiens 6.0
CDC7(CDC7CGP1) CDC7 Homo sapiens 6.0
CDC2 [CDK1(CDK1CGS1)] CDK1 Homo sapiens 6.0
PITSLRE(C11BLGS1) CDK11A Homo sapiens 6.0
CRK7(CD12PHS1) CDK12 Homo sapiens 6.0
CHED(CD13PHS1) CDK13 Homo sapiens 6.0
PFTAIRE1(CD14CGS1) CDK14 Homo sapiens 6.0
PCTAIRE1(CD16SGS1) CDK16 Homo sapiens 6.0
PCTAIRE2(CD17SGS1) CDK17 Homo sapiens 6.0
PCTAIRE3(CD18SGS1) CDK18 Homo sapiens 6.0
CDK11(CD19CGS1) CSNK1E Homo sapiens 6.0
CDK2(CDK2CGS1) CDK2 Homo sapiens 6.0
CDK3(CDK3CGS1) CDK3 Homo sapiens 6.0
CDK4(CDK4CGS1) CDK4 Homo sapiens 6.0
CDK5(CDK5CGS1) CDK5 Homo sapiens 6.0
CDK6(CDK6CGS1) CDK6 Homo sapiens 6.0
CDK7(CDK7CGS1) CDK7 Homo sapiens 6.0
CDK8(CDK8CGS1) CDK8 Homo sapiens 6.0
CDK9(CDK9CGS1) CDK9 Homo sapiens 6.0
CHK1(CHE1CGP1) CHEK1 Homo sapiens 6.0
CHK2(CHE2LGY1) CHEK2 Homo sapiens 6.0
IKKalpha(CHUKLGP1) CHUK Homo sapiens 6.0
CRIK(CIT1LGY1) CIT Homo sapiens 6.0
CLK1(CLK1LGF1) CLK1 Homo sapiens 6.0
CLK2(CLK2LGF1) CLK2 Homo sapiens 6.0
CLK3(CLK3LGY1) CLK3 Homo sapiens 6.0
CLK4(CLK4IGF1) CLK4 Homo sapiens 6.0
FmS [CSFR(CSF1LGC1)] CSF1R Homo sapiens 6.0
CSK(CSK1LGF1) CSK Homo sapiens 6.0
CK1alpha(C1A1PHY1) CSNK1A1 Homo sapiens 6.0
CK1alpha2(C1ALLGI5) CSNK1A1L Homo sapiens 6.0
CK1delta(CS1DLGI1) CSNK1D Homo sapiens 6.0
CK1epsilon(CS1ELGI5) CSNK1E Homo sapiens 6.0
CK1gamma1(C1G1LGI1) CSNK1G1 Homo sapiens 6.0
CK1gamma2(C1G2LGI1) CSNK1G2 Homo sapiens 6.0
CK1gamma3(C1G3LGI5) CSNK1G3 Homo sapiens 6.0
CK2alpha1(C2A1LGF1) CSNK2A1 Homo sapiens 6.0
CK2alpha2(C2A2LGK1) CSNK2A2 Homo sapiens 6.0
DAPK1(DAP1LGF1) DAPK1 Homo sapiens 6.0
DAPK2(DAP2LGF1) DAPK2 Homo sapiens 6.0
DAPK3(DAP3LGP1) DAPK3 Homo sapiens 6.0
DCAMKL3(DCL3LGP1) DCLK3 Homo sapiens 6.0
DMPK(DMPKLGF1) DMPK Homo sapiens 6.0
DYRK1A(DY1ALGP1) DYRK1A Homo sapiens 6.0
DYRK1B(DY1BLHY1) DYRK1B Homo sapiens 6.0
DYRK2(DYR2LGY1) DYRK2 Homo sapiens 6.0
DYRK4(DYR4LHY1) DYRK4 Homo sapiens 6.0
EGFR(EGFRMGB1) EGFR Homo sapiens 6.0
HRI(EIK1CGQ1) EIF2AK1 Homo sapiens 6.0
PKR(EIK2LGY1) EIF2AK2 Homo sapiens 6.0
PERK [PEK(EIK3CGQ1)] EIF2AK3 Homo sapiens 6.0
GCN2(EIK4PHK1) EIF2AK4 Homo sapiens 6.0
EphA1(EPA1LGY1) EPHA1 Homo sapiens 6.0
EphA3(EPA3LGD5) EPHA3 Homo sapiens 6.0
EphA4(EPA4LGF1) EPHA4 Homo sapiens 6.0
EphA5(EPA5MGF1) EPHA5 Homo sapiens 6.0
EphA6(EPA6LGI5) EPHA6 Homo sapiens 6.0
EphA7(EPA7LGF1) EPHA7 Homo sapiens 6.0
EphA8(EPA8LGF1) EPHA8 Homo sapiens 6.0
EphB1(EPB1LGY1) EPHB1 Homo sapiens 6.0
EphB2(EPB2LGY1) EPHB2 Homo sapiens 6.0
EphB3(EPB3LGRJ) EPHB3 Homo sapiens 6.0
EphB4(EPB4LGY1) EPHB4 Homo sapiens 6.0
HER4(ERB4CGF1) ERBB4 Homo sapiens 6.0
IRE1(ERN1PHY1) ERN1 Homo sapiens 6.0
Fer(FER1LGY1) FER Homo sapiens 6.0
Fes(FES1LHY1) FES Homo sapiens 6.0
FGFR3(FGF3LGF1) FGFR3 Homo sapiens 6.0
FGFR4(FGF4LGF1) FGFR4 Homo sapiens 6.0
Fgr(FGR1LGF1) FGR Homo sapiens 6.0
FLT1(FLT1LGC5) FLT1 Homo sapiens 6.0
FLT3(FLT3MGE1) FLT3 Homo sapiens 6.0
FLT4(FLT4LGY1) FLT4 Homo sapiens 6.0
FRK(FRK1LGF1) FRK Homo sapiens 6.0
GAK(GAK1PGF1) GAK Homo sapiens 6.0
RHODK [GRK1(GRK1LGA1)] GRK1 Homo sapiens 6.0
GRK4(GRK4LGRI) GRK4 Homo sapiens 6.0
GRK5(GRK5LGP1) GRK5 Homo sapiens 6.0
GRK6(GRK6LGP1) GRK6 Homo sapiens 6.0
GSK3beta(GS3BLGM1) GSK3B Homo sapiens 6.0
HCK(HCK1LGF1) HCK Homo sapiens 6.0
HIPK1(HIP1LGF1) HIPK1 Homo sapiens 6.0
HIPK2(HIP2LGY1) HIPK2 Homo sapiens 6.0
HIPK4(HIP4LHY1) HIPK4 Homo sapiens 6.0
ICK(ICK1LGP1) CILK1 Homo sapiens 6.0
IGF1R(IGF1LGF1) IGF1R Homo sapiens 6.0
IKKbeta(IKBBLHY1) IKBKB Homo sapiens 6.0
IKKepsilon(IKBELGY1) IKBKE Homo sapiens 6.0
InSR(INSRLGY1) INSR Homo sapiens 6.0
IRR(INSSLGF1) INSRR Homo sapiens 6.0
IRAK3(IRK3PFE1) IRAK3 Homo sapiens 6.0
IRAK4(IRK4LGF1) IRAK4 Homo sapiens 6.0
ITK(ITK1CGF1) ITK Homo sapiens 6.0
JAK3(JAK3LGRG) JAK3 Homo sapiens 6.0
KDR(KDR1CGY1) KDR Homo sapiens 6.0
Kit(KIT1MGC1) KIT Homo sapiens 6.0
LATS1(LAT1LGRJ) LATS1 Homo sapiens 6.0
LATS2(LAT2LGY1) LATS2 Homo sapiens 6.0
Lck(LCK1LGF1) LCK Homo sapiens 6.0
LIMK1(LIM1LGY1) LIMK1 Homo sapiens 6.0
LIMK2(LIM2LGV1) LIMK2 Homo sapiens 6.0
LTK(LTK1LGF1) LTK Homo sapiens 6.0
MEK1 [MAP2K1(M2K1LGF1)] MAP2K1 Homo sapiens 6.0
MKK6 [MAP2K6(M2K6LGF1)] MAP2K6 Homo sapiens 6.0
MLK3(M311LGF1) MAP3K11 Homo sapiens 6.0
DLK(M312CGY1) MAP3K12 Homo sapiens 6.0
LZK(M313LGRJ) MAP3K13 Homo sapiens 6.0
NIK(M314LGP1) MAP3K14 Homo sapiens 6.0
MAP3K7(M315LGP1) MAP3K7 Homo sapiens 6.0
ASK [MAP3K5(M3K5LGA1)] MAP3K5 Homo sapiens 6.0
TAK1(M3K7CHY1) MAP3K7 Homo sapiens 6.0
MLK1(M3K9LGF1) MAP3K9 Homo sapiens 6.0
HPK1(M4K1LGY1) MAP4K1 Homo sapiens 6.0
GCK(M4K2LGY1) GCK Homo sapiens 6.0
HGK [ZC1(M4K4CGP1)] MAP4K4 Homo sapiens 6.0
KHS1(M4K5LGY1) MAP4K5 Homo sapiens 6.0
ERK2(MAP1LGY1) MAPK1 Homo sapiens 6.0
JNK3(MP10LGF2) MAPK10 Homo sapiens 6.0
p38beta(MP11LGI1) MAPK11 Homo sapiens 6.0
p38gamma(MP12LGP1) MAPK12 Homo sapiens 6.0
p38delta(MP13LGP1) MAPK13 Homo sapiens 6.0
p38alpha(MP14LGI1) MAPK14 Homo sapiens 6.0
ERK7(MP15LGY1) MAPK15 Homo sapiens 6.0
ERK1(MAP3LGY1) MAPK3 Homo sapiens 6.0
ERK4(MAP4LGY1) MAPK4 Homo sapiens 6.0
ERK3(MAP6LHY1) MAPK6 Homo sapiens 6.0
JNK1(MAP8LGF1) MAPK8 Homo sapiens 6.0
JNK2(MAP9LGF1) MAPK9 Homo sapiens 6.0
MAPKAPK2(MPK2LGRH) MAPKAPK2 Homo sapiens 6.0
MAPKAPK5(MPK5LGN1) MAPKAPK5 Homo sapiens 6.0
MARK1(MAR1PHY1) MARK1 Homo sapiens 6.0
MARK2(MAR2LGY1) MARK2 Homo sapiens 6.0
MARK3(MAR3LGO5) MARK3 Homo sapiens 6.0
MAST1(MAS1LGE5) MAST1 Homo sapiens 6.0
MAST3(MAS3LGE1) MAST3 Homo sapiens 6.0
MAST4(MAS4LGRD) MAST4 Homo sapiens 6.0
MASTL(MASLLGE1) MASTL Homo sapiens 6.0
MELK(MELKLGF1) MELK Homo sapiens 6.0
Mer(MERTLGF1) MERTK Homo sapiens 6.0
MLKL(MLKLPHY1) MLKL Homo sapiens 6.0
MST4(MST4LGC1) STK26 Homo sapiens 6.0
MUSK(MUSKLGY1) MUSK Homo sapiens 6.0
smMLCK(MYL1LGF1) MYLK Homo sapiens 6.0
skMLCK(MYL2LHY1) MYLK2 Homo sapiens 6.0
caMLCK(MYL3LGF1) MYLK3 Homo sapiens 6.0
MYO3B(MY3BLGA1) MYO3B Homo sapiens 6.0
Nek1(NEK1LGY1) NEK1 Homo sapiens 6.0
Nek11(NE11LGRI) NEK11 Homo sapiens 6.0
Nek2(NEK2LHFA) NEK2 Homo sapiens 6.0
Nek3(NEK3LGRI) NEK3 Homo sapiens 6.0
Nek5(NEK5LGRD) NEK5 Homo sapiens 6.0
Nek8(NEK8LGRI) NEK8 Homo sapiens 6.0
Nek9(NEK9LGF1) NEK9 Homo sapiens 6.0
NLK(NLK1LGI5) NLK Homo sapiens 6.0
TRKA(NTR1LGN1) NTRK1 Homo sapiens 6.0
TRKC(NTR3LGN1) NTRK3 Homo sapiens 6.0
NuaK1(NUA1LGF5) NUAK1 Homo sapiens 6.0
NuaK2(NUA2LHY1) NUAK2 Homo sapiens 6.0
OSR1(OXS1LGY1) OXSR1 Homo sapiens 6.0
PAK4(PAK4CGY1) PAK4 Homo sapiens 6.0
PAK6(PAK6CGY1) PAK6 Homo sapiens 6.0
PAK5(PAK7LGF1) PAK5 Homo sapiens 6.0
PASK(PASKPHY1) PASK Homo sapiens 6.0
PDGFRbeta(PDGBIHC1) PDGFRB Homo sapiens 6.0
PDK1(PDP1LGA1) PDPK1 Homo sapiens 6.0
PhKgamma1(PHG1LHY1) PHKG1 Homo sapiens 6.0
Pim1(PIM1LGP1) PIM1 Homo sapiens 6.0
Pim2(PIM2LHY1) PIM2 Homo sapiens 6.0
Pim3(PIM3LGP1) PIM3 Homo sapiens 6.0
PINK1(PIN1PHRE) PINK1 Homo sapiens 6.0
PKN1 [PRK1(PKN1LGY1)] PKN1 Homo sapiens 6.0
PKN2 [PRK2(PKN2LGG5)] PKN2 Homo sapiens 6.0
PLK1(PLK1LGY1) PLK1 Homo sapiens 6.0
PLK3(PLK3PHY1) PLK3 Homo sapiens 6.0
PLK4(PLK4LGF1) PLK4 Homo sapiens 6.0
CaMK1beta(PNCKLGRI) PNCK Homo sapiens 6.0
AMPKalpha1(PRA1PGF1) PRKAA1 Homo sapiens 6.0
AMPKalpha2(PRA2LGY1) PRKAA2 Homo sapiens 6.0
PKAalpha(PRCALGH1) PRKACA Homo sapiens 6.0
PKAbeta(PRCBLGF1) PRKACB Homo sapiens 6.0
PKAgamma(PRCGLGY1) PRKACG Homo sapiens 6.0
PKCalpha(PRKALGY1) PRKCA Homo sapiens 6.0
PKCbeta(PRKBPHY3) PRKCB Homo sapiens 6.0
PKCdelta(PRKDPFP1) PRKCD Homo sapiens 6.0
PKCepsilon(PRKELHY1) PRKCE Homo sapiens 6.0
PKCeta(PRKHLGRA) PRKCH Homo sapiens 6.0
PKCiota(PRKILGRD) PRKCI Homo sapiens 6.0
PKCtheta(PRKQLGM5) PRKCQ Homo sapiens 6.0
PKCzeta(PRKZLGP1) PRKCZ Homo sapiens 6.0
PKD1(PRD1LHY1) PRKD1 Homo sapiens 6.0
PKD2(PRD2LHY1) PRKD2 Homo sapiens 6.0
PKD3(PRD3LGG5) PRKD3 Homo sapiens 6.0
PKG2(PRG2LHY1) PRKG2 Homo sapiens 6.0
PRKX(PRKXLGH5) PRKX Homo sapiens 6.0
PSKH1(PSH1LGRH) PSKH1 Homo sapiens 6.0
PYK2(PT2BLHF1) PTK2B Homo sapiens 6.0
Brk(PTK6LGY1) PTK6 Homo sapiens 6.0
RIOK2(RIO2LGF1) RIOK2 Homo sapiens 6.0
RIPK1(RIP1PGN1) RIPK1 Homo sapiens 7.7
RIPK2(RIP2LGI1) RIPK2 Homo sapiens 6.0
RIPK3(RIP3IGRI) RIPK3 Homo sapiens 6.0
ROCK1(ROC1LGY1) ROCK1 Homo sapiens 6.0
ROCK2(ROC2LGG1) ROCK2 Homo sapiens 6.0
Ros(ROS1PHY1) ROS1 Homo sapiens 6.0
RSK3(R6A1CGE1) RPS6KA2 Homo sapiens 6.0
RSK1 [p90RSK(R6A2CGE1)] RPS6KA1 Homo sapiens 6.0
MSK2(R6A4LGRJ) RPS6KA4 Homo sapiens 6.0
MSK1(R6A5LGY1) RPS6KA5 Homo sapiens 6.0
RSK4(R6A6LGF1) RPS6KA6 Homo sapiens 6.0
p70S6K(R6B1CGF1) RPS6KB1 Homo sapiens 6.0
SBK(SBK1LGY1) SBK1 Homo sapiens 6.0
SGK2(SGK2LGE5) SGK2 Homo sapiens 6.0
SGK3(SGK3LGY1) SGK3 Homo sapiens 6.0
SIK(SIK1LHY1) SIK1 Homo sapiens 6.0
QIK(SIK2LGY1) SIK2 Homo sapiens 6.0
QSK(SIK3LGP1) SIK3 Homo sapiens 6.0
SLK(SLK1LGRJ) SLK Homo sapiens 6.0
Srm(SRMSLGY1) SRMS Homo sapiens 6.0
SRPK1(SRP1IHRL) SRPK1 Homo sapiens 6.0
SRPK2(SRP2IGRL) SRPK2 Homo sapiens 6.0
MSSK1(SRP3MHRL) SRPK3 Homo sapiens 6.0
MST3(ST24LGC1) STK24 Homo sapiens 6.0
MST2(STK3LGF1) STK3 Homo sapiens 6.0
YANK1(S32APHY1) STK32A Homo sapiens 6.0
YANK2(S32BLGY2) STK32B Homo sapiens 6.0
YANK3(S32CLGI1) STK32C Homo sapiens 6.0
STK33(ST33LGF1) STK33 Homo sapiens 6.0
STLK3(ST39LGRJ) STK39 Homo sapiens 6.0
MST1(STK4LGF1) STK4 Homo sapiens 6.0
STLK5(STRAPHD1) STRADA Homo sapiens 6.0
Syk(SYK1LHY1) SYK Homo sapiens 6.0
TAO2(TAO2LGF1) TAOK2 Homo sapiens 6.0
TAO3(TAO3LGY1) TAOK3 Homo sapiens 6.0
TBK1(TBK1CGF1) TBK1 Homo sapiens 6.0
TEC(TEC1CGD1) TEC Homo sapiens 6.0
TESK2(TES2LGRL) TESK2 Homo sapiens 6.0
TGFbetaR1(TGF1LGF1) TGFBR1 Homo sapiens 6.0
TGFbetaR2(TGF2LGY1) TGFBR2 Homo sapiens 6.0
TLK1(TLK1LGP1) TLK1 Homo sapiens 6.0
TNIK [ZC2(TNIKLGF1)] TNIK Homo sapiens 6.0
Tnk1(TNK1LGY1) TNK1 Homo sapiens 6.0
Ack(TNK2LGF1) TNK2 Homo sapiens 6.0
HH498(TNNILGY1) TNNI3K Homo sapiens 6.0
TSSK1(TS1BLGP1) TSSK1B Homo sapiens 6.0
TXK(TXK1CGD5) TXK Homo sapiens 6.0
Tyk2(TYK2LGF1) TYK2 Homo sapiens 6.0
ULK1(ULK1LGF1) ULK1 Homo sapiens 6.0
ULK2(ULK2LGY1) ULK2 Homo sapiens 6.0
ULK3(ULK3LGF1) ULK3 Homo sapiens 6.0
VRK1(VRK1LGRI) VRK1 Homo sapiens 6.0
VRK2(VRK2LGRI) VRK2 Homo sapiens 6.0
Wee1(WEE1LGF1) WEE1 Homo sapiens 6.0
ZAK(ZAK1LGY1) MAP3K20 Homo sapiens 6.0
HUNK(HUNKLGRN) HUNK Homo sapiens 6.0
SgK085(SG85LGY1) MYLK4 Homo sapiens 6.0
Wee1B(WE1BLGF1) WEE2 Homo sapiens 6.0
SgK110(SG10LGF1) SBK3 Homo sapiens 6.0
PI3KCA(PI3ACGR1) PIK3CA Homo sapiens 6.0
CDK11A(C11ALGS1) CDK11A Homo sapiens 6.0
PIK3CB(PI3BCGRK) PIK3CB Homo sapiens 6.0
PI3KCD(PI3DCGRK) PIK3CD Homo sapiens 6.0
BRD4(BRD4LGRC) BRD4 Homo sapiens 6.0
BRDT(BRDTLGRC) BRDT Homo sapiens 6.0
 

TP-030n

Conclusion: Clean panel

Target protein HGNC name Species pIC50
Abl(ABL1IHY1) ABL1 Homo sapiens 6.0
Arg(ABL2LGF1) ABL2 Homo sapiens 6.0
ALK2(ACV1LGF1) ACVR1 Homo sapiens 6.0
ACtR2(AC2ALGE1) ACVR2A Homo sapiens 6.0
ALK1(ACL1LGF1) ACVRL1 Homo sapiens 6.0
BARK1 [GRK2(ADR1LGG5)] GRK2 Homo sapiens 6.0
BARK2 [GRK3(ADR2LGG5)] GRK3 Homo sapiens 6.0
Akt2 [PKBbeta(AKT2CGY1)] AKT2 Homo sapiens 6.0
Akt3 [PKBgamma(AKT3LGY1)] AKT3 Homo sapiens 6.0
ALK(ALK1LGY1) ALK Homo sapiens 6.0
SgK288(ANK1LGRL) ANKK1 Homo sapiens 6.0
AurA [Aur2(AURALGF1)] AURKA Homo sapiens 6.0
AurB [Aur1(AURBPGE1)] AURKB Homo sapiens 6.0
Axl(AXL1LGY1) AXL Homo sapiens 6.0
BLK(BLK1CGF1) BLK Homo sapiens 6.0
BIKE(BM2KLGY1) BMP2K Homo sapiens 6.0
BMPR1A(BM1APHRG) BMPR1A Homo sapiens 6.0
BMPR1B(BM1BLGF1) BMPR1B Homo sapiens 6.0
BMPR2(BMR2LGN1) BMPR2 Homo sapiens 6.0
Etk [BMX(BMX1CGF1)] BMX Homo sapiens 6.0
BRAF(BRAFLGY1) BRAF Homo sapiens 6.0
BRSK1(BRS1LGA1) BRSK1 Homo sapiens 6.0
BTK(BTK1CGF1) BTK Homo sapiens 6.0
Bub1(BUB1LGRL) BUB1 Homo sapiens 6.0
CaMK1gamma(CA1GLGN1) CAMK1G Homo sapiens 6.0
CaMK4(CAM4LGY1) CAMK4 Homo sapiens 6.0
CASK(CASKLGY1) CASK Homo sapiens 6.0
MRCKalpha(CD4ALGY1) CDC42BPA Homo sapiens 6.0
DMPK2(CD4GLGRD) EPHB1 Homo sapiens 6.0
CDC7(CDC7CGP1) CDC7 Homo sapiens 6.0
CDC2 [CDK1(CDK1CGS1)] CDK1 Homo sapiens 6.0
PITSLRE(C11BLGS1) CDK11A Homo sapiens 6.0
CRK7(CD12PHS1) CDK12 Homo sapiens 6.0
CHED(CD13PHS1) CDK13 Homo sapiens 6.0
PFTAIRE1(CD14CGS1) CDK14 Homo sapiens 6.0
PCTAIRE1(CD16SGS1) CDK16 Homo sapiens 6.0
PCTAIRE2(CD17SGS1) CDK17 Homo sapiens 6.0
PCTAIRE3(CD18SGS1) CDK18 Homo sapiens 6.0
CDK11(CD19CGS1) CSNK1E Homo sapiens 6.0
CDK2(CDK2CGS1) CDK2 Homo sapiens 6.0
CDK3(CDK3CGS1) CDK3 Homo sapiens 6.0
CDK4(CDK4CGS1) CDK4 Homo sapiens 6.0
CDK5(CDK5CGS1) CDK5 Homo sapiens 6.0
CDK6(CDK6CGS1) CDK6 Homo sapiens 6.0
CDK7(CDK7CGS1) CDK7 Homo sapiens 6.0
CDK8(CDK8CGS1) CDK8 Homo sapiens 6.0
CDK9(CDK9CGS1) CDK9 Homo sapiens 6.0
CHK1(CHE1CGP1) CHEK1 Homo sapiens 6.0
CHK2(CHE2LGY1) CHEK2 Homo sapiens 6.0
IKKalpha(CHUKLGP1) CHUK Homo sapiens 6.0
CRIK(CIT1LGY1) CIT Homo sapiens 6.0
CLK1(CLK1LGF1) CLK1 Homo sapiens 6.0
CLK2(CLK2LGF1) CLK2 Homo sapiens 6.0
CLK3(CLK3LGY1) CLK3 Homo sapiens 6.0
CLK4(CLK4IGF1) CLK4 Homo sapiens 6.0
FmS [CSFR(CSF1LGC1)] CSF1R Homo sapiens 6.0
CSK(CSK1LGF1) CSK Homo sapiens 6.0
CK1alpha(C1A1PHY1) CSNK1A1 Homo sapiens 6.0
CK1alpha2(C1ALLGI5) CSNK1A1L Homo sapiens 6.0
CK1delta(CS1DLGI1) CSNK1D Homo sapiens 6.0
CK1epsilon(CS1ELGI5) CSNK1E Homo sapiens 6.0
CK1gamma1(C1G1LGI1) CSNK1G1 Homo sapiens 6.0
CK1gamma2(C1G2LGI1) CSNK1G2 Homo sapiens 6.0
CK1gamma3(C1G3LGI5) CSNK1G3 Homo sapiens 6.0
CK2alpha1(C2A1LGF1) CSNK2A1 Homo sapiens 6.0
CK2alpha2(C2A2LGK1) CSNK2A2 Homo sapiens 6.0
DAPK1(DAP1LGF1) DAPK1 Homo sapiens 6.0
DAPK2(DAP2LGF1) DAPK2 Homo sapiens 6.0
DAPK3(DAP3LGP1) DAPK3 Homo sapiens 6.0
DCAMKL3(DCL3LGP1) DCLK3 Homo sapiens 6.0
DMPK(DMPKLGF1) DMPK Homo sapiens 6.0
DYRK1A(DY1ALGP1) DYRK1A Homo sapiens 6.0
DYRK1B(DY1BLHY1) DYRK1B Homo sapiens 6.0
DYRK2(DYR2LGY1) DYRK2 Homo sapiens 6.0
DYRK4(DYR4LHY1) DYRK4 Homo sapiens 6.0
EGFR(EGFRMGB1) EGFR Homo sapiens 6.0
HRI(EIK1CGQ1) EIF2AK1 Homo sapiens 6.0
PKR(EIK2LGY1) EIF2AK2 Homo sapiens 6.0
PERK [PEK(EIK3CGQ1)] EIF2AK3 Homo sapiens 6.0
GCN2(EIK4PHK1) EIF2AK4 Homo sapiens 6.0
EphA1(EPA1LGY1) EPHA1 Homo sapiens 6.0
EphA3(EPA3LGD5) EPHA3 Homo sapiens 6.0
EphA4(EPA4LGF1) EPHA4 Homo sapiens 6.0
EphA5(EPA5MGF1) EPHA5 Homo sapiens 6.0
EphA6(EPA6LGI5) EPHA6 Homo sapiens 6.0
EphA7(EPA7LGF1) EPHA7 Homo sapiens 6.0
EphA8(EPA8LGF1) EPHA8 Homo sapiens 6.0
EphB1(EPB1LGY1) EPHB1 Homo sapiens 6.0
EphB2(EPB2LGY1) EPHB2 Homo sapiens 6.0
EphB3(EPB3LGRJ) EPHB3 Homo sapiens 6.0
EphB4(EPB4LGY1) EPHB4 Homo sapiens 6.0
HER4(ERB4CGF1) ERBB4 Homo sapiens 6.0
IRE1(ERN1PHY1) ERN1 Homo sapiens 6.0
Fer(FER1LGY1) FER Homo sapiens 6.0
Fes(FES1LHY1) FES Homo sapiens 6.0
FGFR3(FGF3LGF1) FGFR3 Homo sapiens 6.0
FGFR4(FGF4LGF1) FGFR4 Homo sapiens 6.0
Fgr(FGR1LGF1) FGR Homo sapiens 6.0
FLT1(FLT1LGC5) FLT1 Homo sapiens 6.0
FLT3(FLT3MGE1) FLT3 Homo sapiens 6.0
FLT4(FLT4LGY1) FLT4 Homo sapiens 6.0
FRK(FRK1LGF1) FRK Homo sapiens 6.0
GAK(GAK1PGF1) GAK Homo sapiens 6.0
RHODK [GRK1(GRK1LGA1)] GRK1 Homo sapiens 6.0
GRK4(GRK4LGRI) GRK4 Homo sapiens 6.0
GRK5(GRK5LGP1) GRK5 Homo sapiens 6.0
GRK6(GRK6LGP1) GRK6 Homo sapiens 6.0
GSK3beta(GS3BLGM1) GSK3B Homo sapiens 6.0
HCK(HCK1LGF1) HCK Homo sapiens 6.0
HIPK1(HIP1LGF1) HIPK1 Homo sapiens 6.0
HIPK2(HIP2LGY1) HIPK2 Homo sapiens 6.0
HIPK4(HIP4LHY1) HIPK4 Homo sapiens 6.0
ICK(ICK1LGP1) CILK1 Homo sapiens 6.0
IGF1R(IGF1LGF1) IGF1R Homo sapiens 6.0
IKKbeta(IKBBLHY1) IKBKB Homo sapiens 6.0
IKKepsilon(IKBELGY1) IKBKE Homo sapiens 6.0
InSR(INSRLGY1) INSR Homo sapiens 6.0
IRR(INSSLGF1) INSRR Homo sapiens 6.0
IRAK3(IRK3PFE1) IRAK3 Homo sapiens 6.0
IRAK4(IRK4LGF1) IRAK4 Homo sapiens 6.0
ITK(ITK1CGF1) ITK Homo sapiens 6.0
JAK3(JAK3LGRG) JAK3 Homo sapiens 6.0
KDR(KDR1CGY1) KDR Homo sapiens 6.0
Kit(KIT1MGC1) KIT Homo sapiens 6.0
LATS2(LAT2LGY1) LATS2 Homo sapiens 6.0
Lck(LCK1LGF1) LCK Homo sapiens 6.0
LIMK1(LIM1LGY1) LIMK1 Homo sapiens 6.0
LIMK2(LIM2LGV1) LIMK2 Homo sapiens 6.0
LTK(LTK1LGF1) LTK Homo sapiens 6.0
MEK1 [MAP2K1(M2K1LGF1)] MAP2K1 Homo sapiens 6.0
MKK6 [MAP2K6(M2K6LGF1)] MAP2K6 Homo sapiens 6.0
MLK3(M311LGF1) MAP3K11 Homo sapiens 6.0
DLK(M312CGY1) MAP3K12 Homo sapiens 6.0
LZK(M313LGRJ) MAP3K13 Homo sapiens 6.0
NIK(M314LGP1) MAP3K14 Homo sapiens 6.0
MAP3K7(M315LGP1) MAP3K7 Homo sapiens 6.0
ASK [MAP3K5(M3K5LGA1)] MAP3K5 Homo sapiens 6.0
TAK1(M3K7CHY1) MAP3K7 Homo sapiens 6.0
MLK1(M3K9LGF1) MAP3K9 Homo sapiens 6.0
HPK1(M4K1LGY1) MAP4K1 Homo sapiens 6.0
GCK(M4K2LGY1) GCK Homo sapiens 6.0
KHS1(M4K5LGY1) MAP4K5 Homo sapiens 6.0
ERK2(MAP1LGY1) MAPK1 Homo sapiens 6.0
JNK3(MP10LGF2) MAPK10 Homo sapiens 6.0
p38beta(MP11LGI1) MAPK11 Homo sapiens 6.0
p38gamma(MP12LGP1) MAPK12 Homo sapiens 6.0
p38delta(MP13LGP1) MAPK13 Homo sapiens 6.0
p38alpha(MP14LGI1) MAPK14 Homo sapiens 6.0
ERK7(MP15LGY1) MAPK15 Homo sapiens 6.0
ERK1(MAP3LGY1) MAPK3 Homo sapiens 6.0
ERK3(MAP6LHY1) MAPK6 Homo sapiens 6.0
JNK1(MAP8LGF1) MAPK8 Homo sapiens 6.0
JNK2(MAP9LGF1) MAPK9 Homo sapiens 6.0
MAPKAPK2(MPK2LGRH) MAPKAPK2 Homo sapiens 6.0
MAPKAPK5(MPK5LGN1) MAPKAPK5 Homo sapiens 6.0
MARK1(MAR1PHY1) MARK1 Homo sapiens 6.0
MARK2(MAR2LGY1) MARK2 Homo sapiens 6.0
MARK3(MAR3LGO5) MARK3 Homo sapiens 6.0
MAST1(MAS1LGE5) MAST1 Homo sapiens 6.0
MAST3(MAS3LGE1) MAST3 Homo sapiens 6.0
MAST4(MAS4LGRD) MAST4 Homo sapiens 6.0
MASTL(MASLLGE1) MASTL Homo sapiens 6.0
MELK(MELKLGF1) MELK Homo sapiens 6.0
Mer(MERTLGF1) MERTK Homo sapiens 6.0
MLKL(MLKLPHY1) MLKL Homo sapiens 6.0
MST4(MST4LGC1) STK26 Homo sapiens 6.0
MUSK(MUSKLGY1) MUSK Homo sapiens 6.0
smMLCK(MYL1LGF1) MYLK Homo sapiens 6.0
skMLCK(MYL2LHY1) MYLK2 Homo sapiens 6.0
caMLCK(MYL3LGF1) MYLK3 Homo sapiens 6.0
MYO3B(MY3BLGA1) MYO3B Homo sapiens 6.0
Nek1(NEK1LGY1) NEK1 Homo sapiens 6.0
Nek11(NE11LGRI) NEK11 Homo sapiens 6.0
Nek2(NEK2LHFA) NEK2 Homo sapiens 6.0
Nek3(NEK3LGRI) NEK3 Homo sapiens 6.0
Nek5(NEK5LGRD) NEK5 Homo sapiens 6.0
Nek9(NEK9LGF1) NEK9 Homo sapiens 6.0
NLK(NLK1LGI5) NLK Homo sapiens 6.0
TRKA(NTR1LGN1) NTRK1 Homo sapiens 6.0
TRKC(NTR3LGN1) NTRK3 Homo sapiens 6.0
NuaK1(NUA1LGF5) NUAK1 Homo sapiens 6.0
NuaK2(NUA2LHY1) NUAK2 Homo sapiens 6.0
OSR1(OXS1LGY1) OXSR1 Homo sapiens 6.0
PAK4(PAK4CGY1) PAK4 Homo sapiens 6.0
PAK6(PAK6CGY1) PAK6 Homo sapiens 6.0
PAK5(PAK7LGF1) PAK5 Homo sapiens 6.0
PASK(PASKPHY1) PASK Homo sapiens 6.0
PDGFRbeta(PDGBIHC1) PDGFRB Homo sapiens 6.0
PDK1(PDP1LGA1) PDPK1 Homo sapiens 6.0
PhKgamma1(PHG1LHY1) PHKG1 Homo sapiens 6.0
Pim1(PIM1LGP1) PIM1 Homo sapiens 6.0
Pim2(PIM2LHY1) PIM2 Homo sapiens 6.0
Pim3(PIM3LGP1) PIM3 Homo sapiens 6.0
PINK1(PIN1PHRE) PINK1 Homo sapiens 6.0
PKN1 [PRK1(PKN1LGY1)] PKN1 Homo sapiens 6.0
PLK1(PLK1LGY1) PLK1 Homo sapiens 6.0
PLK3(PLK3PHY1) PLK3 Homo sapiens 6.0
PLK4(PLK4LGF1) PLK4 Homo sapiens 6.0
CaMK1beta(PNCKLGRI) PNCK Homo sapiens 6.0
AMPKalpha1(PRA1PGF1) PRKAA1 Homo sapiens 6.0
AMPKalpha2(PRA2LGY1) PRKAA2 Homo sapiens 6.0
PKAalpha(PRCALGH1) PRKACA Homo sapiens 6.0
PKAbeta(PRCBLGF1) PRKACB Homo sapiens 6.0
PKAgamma(PRCGLGY1) PRKACG Homo sapiens 6.0
PKCalpha(PRKALGY1) PRKCA Homo sapiens 6.0
PKCbeta(PRKBPHY3) PRKCB Homo sapiens 6.0
PKCdelta(PRKDPFP1) PRKCD Homo sapiens 6.0
PKCepsilon(PRKELHY1) PRKCE Homo sapiens 6.0
PKCeta(PRKHLGRA) PRKCH Homo sapiens 6.0
PKCiota(PRKILGRD) PRKCI Homo sapiens 6.0
PKCtheta(PRKQLGM5) PRKCQ Homo sapiens 6.0
PKCzeta(PRKZLGP1) PRKCZ Homo sapiens 6.0
PKD1(PRD1LHY1) PRKD1 Homo sapiens 6.0
PKD2(PRD2LHY1) PRKD2 Homo sapiens 6.0
PKD3(PRD3LGG5) PRKD3 Homo sapiens 6.0
PKG2(PRG2LHY1) PRKG2 Homo sapiens 6.0
PRKX(PRKXLGH5) PRKX Homo sapiens 6.0
PSKH1(PSH1LGRH) PSKH1 Homo sapiens 6.0
PYK2(PT2BLHF1) PTK2B Homo sapiens 6.0
Brk(PTK6LGY1) PTK6 Homo sapiens 6.0
RIOK2(RIO2LGF1) RIOK2 Homo sapiens 6.0
RIPK1(RIP1PGN1) RIPK1 Homo sapiens 6.0
RIPK2(RIP2LGI1) RIPK2 Homo sapiens 6.0
RIPK3(RIP3IGRI) RIPK3 Homo sapiens 6.0
ROCK1(ROC1LGY1) ROCK1 Homo sapiens 6.0
ROCK2(ROC2LGG1) ROCK2 Homo sapiens 6.0
Ros(ROS1PHY1) ROS1 Homo sapiens 6.0
RSK3(R6A1CGE1) RPS6KA2 Homo sapiens 6.0
RSK1 [p90RSK(R6A2CGE1)] RPS6KA1 Homo sapiens 6.0
MSK2(R6A4LGRJ) RPS6KA4 Homo sapiens 6.0
MSK1(R6A5LGY1) RPS6KA5 Homo sapiens 6.0
RSK4(R6A6LGF1) RPS6KA6 Homo sapiens 6.0
p70S6K(R6B1CGF1) RPS6KB1 Homo sapiens 6.0
SBK(SBK1LGY1) SBK1 Homo sapiens 6.0
SGK2(SGK2LGE5) SGK2 Homo sapiens 6.0
SGK3(SGK3LGY1) SGK3 Homo sapiens 6.0
QIK(SIK2LGY1) SIK2 Homo sapiens 6.0
QSK(SIK3LGP1) SIK3 Homo sapiens 6.0
SLK(SLK1LGRJ) SLK Homo sapiens 6.0
Srm(SRMSLGY1) SRMS Homo sapiens 6.0
SRPK1(SRP1IHRL) SRPK1 Homo sapiens 6.0
SRPK2(SRP2IGRL) SRPK2 Homo sapiens 6.0
MSSK1(SRP3MHRL) SRPK3 Homo sapiens 6.0
MST3(ST24LGC1) STK24 Homo sapiens 6.0
MST2(STK3LGF1) STK3 Homo sapiens 6.0
YANK1(S32APHY1) STK32A Homo sapiens 6.0
YANK2(S32BLGY2) STK32B Homo sapiens 6.0
YANK3(S32CLGI1) STK32C Homo sapiens 6.0
STK33(ST33LGF1) STK33 Homo sapiens 6.0
MST1(STK4LGF1) STK4 Homo sapiens 6.0
STLK5(STRAPHD1) STRADA Homo sapiens 6.0
Syk(SYK1LHY1) SYK Homo sapiens 6.0
TAO2(TAO2LGF1) TAOK2 Homo sapiens 6.0
TAO3(TAO3LGY1) TAOK3 Homo sapiens 6.0
TBK1(TBK1CGF1) TBK1 Homo sapiens 6.0
TEC(TEC1CGD1) TEC Homo sapiens 6.0
TESK2(TES2LGRL) TESK2 Homo sapiens 6.0
TGFbetaR1(TGF1LGF1) TGFBR1 Homo sapiens 6.0
TGFbetaR2(TGF2LGY1) TGFBR2 Homo sapiens 6.0
TLK1(TLK1LGP1) TLK1 Homo sapiens 6.0
TNIK [ZC2(TNIKLGF1)] TNIK Homo sapiens 6.0
Tnk1(TNK1LGY1) TNK1 Homo sapiens 6.0
Ack(TNK2LGF1) TNK2 Homo sapiens 6.0
HH498(TNNILGY1) TNNI3K Homo sapiens 6.0
TSSK1(TS1BLGP1) TSSK1B Homo sapiens 6.0
TXK(TXK1CGD5) TXK Homo sapiens 6.0
Tyk2(TYK2LGF1) TYK2 Homo sapiens 6.0
ULK1(ULK1LGF1) ULK1 Homo sapiens 6.0
ULK2(ULK2LGY1) ULK2 Homo sapiens 6.0
ULK3(ULK3LGF1) ULK3 Homo sapiens 6.0
VRK1(VRK1LGRI) VRK1 Homo sapiens 6.0
VRK2(VRK2LGRI) VRK2 Homo sapiens 6.0
Wee1(WEE1LGF1) WEE1 Homo sapiens 6.0
ZAK(ZAK1LGY1) MAP3K20 Homo sapiens 6.0
HUNK(HUNKLGRN) HUNK Homo sapiens 6.0
SgK085(SG85LGY1) MYLK4 Homo sapiens 6.0
Wee1B(WE1BLGF1) WEE2 Homo sapiens 6.0
SgK110(SG10LGF1) SBK3 Homo sapiens 6.0
PI3KCA(PI3ACGR1) PIK3CA Homo sapiens 6.0
CDK11A(C11ALGS1) CDK11A Homo sapiens 6.0
PIK3CB(PI3BCGRK) PIK3CB Homo sapiens 6.0
PI3KCD(PI3DCGRK) PIK3CD Homo sapiens 6.0
BRD4(BRD4LGRC) BRD4 Homo sapiens 6.0
BRDT(BRDTLGRC) BRDT Homo sapiens 6.0
AAK1(AAK1LGF1) AAK1 Homo sapiens 6.0
ALK4(AC1BLGF1) ACVR1B Homo sapiens 6.0
Akt1 [PKBalpha(AKT1PHFB)] AKT1 Homo sapiens 6.0
CaMK1alpha(CAM1LGT5) CAMK1 Homo sapiens 6.0
CaMK1delta(CA1DLGT5) CAMK1D Homo sapiens 6.0
CaMK2alpha(CA2ACGT1) CAMK2A Homo sapiens 6.0
CaMK2beta(CA2BCGT1) CAMK2B Homo sapiens 6.0
CaMK2delta(CA2DCGT1) CAMK2D Homo sapiens 6.0
CaMK2gamma(CA2GLGT5) CAMK2G Homo sapiens 6.0
CAMKK1(CAK1LGT5) CAMKK1 Homo sapiens 6.0
CAMKK2(CAK2LGT5) CAMKK2 Homo sapiens 6.0
CDKL1(CDL1LGT1) CDKL1 Homo sapiens 6.0
DDR1(DDR1LGF1) DDR1 Homo sapiens 6.0
EphA2(EPA2LGY1) EPHA2 Homo sapiens 6.0
FGFR1(FGF1LGF1) FGFR1 Homo sapiens 6.0
FGFR2(FGF2LGF1) FGFR2 Homo sapiens 6.0
Fyn(FYN1LGF5) FYN Homo sapiens 6.0
GSK3alpha(GS3ALGK1) GSK3A Homo sapiens 6.0
HIPK3(HIP3LGF1) HIPK3 Homo sapiens 6.0
IRAK1(IRK1LGF1) IRAK1 Homo sapiens 6.0
JAK2(JAK2LGF1) JAK2 Homo sapiens 6.0
LRRK2(LRR2PGF1) LRRK2 Homo sapiens 6.0
Lyn(LYN1LGF1) LYN Homo sapiens 6.0
MEK2 [MAP2K2(M2K2LGF1)] MAP2K2 Homo sapiens 6.0
MAP2K7(M2K7CGRI) MAP2K7 Homo sapiens 6.0
MEKK2 [MAP3K2(M3K2LGF1)] MAP3K2 Homo sapiens 6.0
ERK5(MAP7LGF1) MAPK7 Homo sapiens 6.0
Met(MEK1LGF1) MET Homo sapiens 6.0
MINK [ZC3(MIN1LGF1)] MINK1 Homo sapiens 6.0
Ron(MST1MGY1) MST1R Homo sapiens 6.0
MYO3A(MY3ALGRI) MYO3A Homo sapiens 6.0
PhKgamma2(PHG2LGF1) PHKG2 Homo sapiens 6.0
PKCgamma(PRKGLGP1) PRKCG Homo sapiens 6.0
PKG1(PRG1LFP1) PRKG1 Homo sapiens 6.0
FAK(PTK2LGF1) PTK2 Homo sapiens 6.0
Ret(RET1LGF1) RET Homo sapiens 6.0
ANKRD3(RIP4LGN1) RIPK4 Homo sapiens 6.0
RSK2(R6A3CGE1) RPS6KA3 Homo sapiens 6.0
SGK1(SGK1LGF1) SGK1 Homo sapiens 6.0
Src(SRC1LGF5) SRC Homo sapiens 6.0
MPSK1(ST16LGF1) STK16 Homo sapiens 6.0
YSK1(ST25LHY1) STK25 Homo sapiens 6.0
NDR1(ST38LGF1) STK38 Homo sapiens 6.0
NDR2(S38LLGF1) STK38L Homo sapiens 6.0
TAO1(TAO1LGF1) TAOK1 Homo sapiens 6.0
TIE2(TEK1LGF1) TEK Homo sapiens 6.0
TESK1(TES1LGRA) TESK1 Homo sapiens 6.0
Trb1(TRI1PARP) TRIB1 Homo sapiens 6.0
TSSK3(TSS3LGRM) TSSK3 Homo sapiens 6.0
Tyro3 [Sky(TYR3LGY1)] TYRO3 Homo sapiens 6.0
Yes(YES1LGF1) YES1 Homo sapiens 6.0
ZAP70(ZAP7LGP1) ZAP70 Homo sapiens 6.0
BRD2(BRD2LHRC) BRD2 Homo sapiens 6.0