Physicochemical properties of probe BAY-474 and control BAY-827
| BAY-474 | |
|---|---|
| TPSA | 88 Å2 |
| log D (pH 7.5) | 1.7 |
| BAY-827 | |
|---|---|
| TPSA | 88 Å2 |
| Calculated log D (pH 7.5) | 7.8 |
Solubility
| BAY-474: |
aqueous pH 6.5: 1.2 mg/L
|
| BAY-827: |
water pH 6.5 : 17 mg/L
|