Physicochemical properties of probe BAY-6672 and control BAY-403
| BAY-6672 | |
|---|---|
| log D (pH 7.5) | 2.3 |
| Ligand-lipophilicity efficiency (LLE) | 5.5 |
| Binding efficiency index (BEI) | 17.0 |
| BAY-403 | |
|---|---|
| log D (pH 7.5) | 1.7 |
| Ligand-lipophilicity efficiency (LLE) | 4.0 |
| Binding efficiency index (BEI) | 12.0 |
Solubility
| BAY-6672: |
aqueous solution pH 6.5: 100 mg/L
|
| BAY-403: |
aqueous solution pH 6.5: 493 mg/L
|